SCHEMBL185085

SCHEMBL185085

COc1ccc(N(C)c2ccc(CNC(=O)C3(NC(=O)Oc4cncnc4)CC3)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 1/20 0.47
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
TRPV1 Q8NER1 2/20 0.41
PPIB P23284 1/20 0.41
FAAH O00519 1/20 0.41
RAB9A P51151 3/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
F10 P00742 1/20 0.39
NPC1 O15118 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGDS O60760 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL187120 0.91 BDKRB1 (0.50) BDKRB1TRPV1PPIBFAAHRAB9A
SCHEMBL2806959 0.89 BDKRB1 (0.59) BDKRB1ALDH1A1SMN1; SMN2PPIBRAB9A
SCHEMBL14856425 0.88 BDKRB1 (0.48) BDKRB1ALDH1A1SMN1; SMN2TRPV1FAAH
SCHEMBL185880 0.85 BDKRB1 (0.47) BDKRB1TRPV1FAAHRAB9ACYP3A4
SCHEMBL185841 0.84 BDKRB1 (0.46) BDKRB1ALDH1A1SMN1; SMN2TRPV1FAAH
SCHEMBL185457 0.82 BDKRB1 (0.49) BDKRB1TRPV1FAAHRAB9ANPC1
SCHEMBL754425 0.81 PPARD (0.44) BDKRB1ALDH1A1SMN1; SMN2TRPV1FAAH
SCHEMBL13128621 0.79 BDKRB1 (0.53) BDKRB1ALDH1A1SMN1; SMN2PPIBRAB9A
SCHEMBL765812 0.79 BDKRB1 (0.63) BDKRB1ALDH1A1SMN1; SMN2RAB9ACYP1A2
SCHEMBL756449 0.78 BDKRB1 (0.46) BDKRB1ALDH1A1SMN1; SMN2FAAHCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401256-B1 Compounds as bradykinin B1 antagonists BOEHRINGER INGELHEIM INT (DE) 2013-04-17 EP disclosed
EP-2401256-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-01-04 EP disclosed
WO-2010097372-A1 COMPOUNDS AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed