SCHEMBL18530342

SCHEMBL18530342

CCc1cccc(C(C(N)=O)C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.46
EPHX1 P07099 4/20 0.44
BCL2 P10415 1/20 0.44
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CTSB P07858 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
SIGMAR1 Q99720 2/20 0.40
MAPT P10636 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682035 0.86 PTGS2 (0.51) PTGS2EPHX1BCL2TSHRMAPK1
SCHEMBL28252817 0.83 ENPP2 (0.48) EPHX1TSHRCYP3A4CYP2D6SMN1; SMN2
SCHEMBL11077922 0.81 ALDH1A1 (0.44) PTGS2EPHX1BCL2TSHRMAPK1
SCHEMBL11080208 0.79 EPHX1 (0.44) PTGS2EPHX1BCL2TSHRMAPK1
SCHEMBL38659679 0.79 PTGS2 (0.51) PTGS2BCL2TDP1CTSBCYP2D6
SCHEMBL7556579 0.77 EPHX1 (0.71) PTGS2EPHX1BCL2CTSB
SCHEMBL18242200 0.77 PTGS2 (0.41) PTGS2BCL2TSHRMAPK1TDP1
SCHEMBL2552458 0.76 LMNA (0.53) PTGS2BCL2TSHRMAPK1CTSB
SCHEMBL2552459 0.76 LMNA (0.53) PTGS2BCL2TSHRMAPK1CTSB
SCHEMBL3674499 0.76 PTGS2 (0.69) PTGS2BCL2TSHRMAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026027-B Substituted malonamide compounds and their use as antibacterial agents 邱浩杰 2020-10-02 CN disclosed
EP-3331852-A1 SUBSTITUTED MALONAMIDES AND THEIR USE AS ANTIBACTERIAL DRUGS National Taiwan University (TW) 2018-06-13 EP disclosed
WO-2017028745-A1 SUBSTITUTED MALONAMIDES AND THEIR USE AS ANTIBACTERIAL DRUGS SHIAU CHUNG-WAI (CN) 2017-02-23 WO disclosed