SCHEMBL18534818

SCHEMBL18534818

N=Cc1c(N)cc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 0.39
TSHR P16473 7/20 0.39
TP53 P04637 2/20 0.39
ALDH1A1 P00352 8/20 0.36
GAA P10253 1/20 0.36
ALOX15 P16050 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
HSD17B10 Q99714 4/20 0.33
RECQL P46063 3/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 1/20 0.33
HPGD P15428 3/20 0.32
THRB P10828 3/20 0.32
CASP1 P29466 2/20 0.32
ALOX12 P18054 2/20 0.32
MAPK1 P28482 2/20 0.32
RIPK1 Q13546 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21600440 0.83 ALDH1A1 (0.45) CYP3A4TSHRTP53ALDH1A1ALOX15
SCHEMBL17739137 0.78 CYP3A4 (0.33) CYP3A4TSHRTP53ALDH1A1ALOX15
SCHEMBL18534544 0.78 CYP3A4 (0.33) CYP3A4TSHRTP53ALDH1A1ALOX15
SCHEMBL16627925 0.73 TSHR (0.50) CYP3A4TSHRALDH1A1ALOX15SMN1; SMN2
SCHEMBL17739390 0.72 LMNA (0.39) CYP3A4TP53ALDH1A1LMNAHTT
SCHEMBL17739398 0.72 TAAR1 (0.33) TDP1RECQLTHRBMEN1HTR2C
SCHEMBL17739108 0.71 GABRA1 (0.37) CYP3A4
Guanidine SCHEMBL10918002 0.71 THRB (0.44) CYP3A4TSHRTP53ALDH1A1ALOX15
SCHEMBL17738734 0.69 GABRA1 (0.32)
SCHEMBL17739334 0.69 GABRA1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763990-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2017-02-22 EP disclosed