SCHEMBL18536009

SCHEMBL18536009

CCCCc1cc(C)c(C)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SKP2 Q13309 1/20 0.50
ALDH1A1 P00352 2/20 0.45
CYP1A2 P05177 1/20 0.45
ALOX15 P16050 1/20 0.45
CASP7 P55210 1/20 0.45
HIF1A Q16665 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPK1 P28482 2/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42
NOS2 P35228 1/20 0.40
TLR8 Q9NR97 2/20 0.40
TYR P14679 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL833088 0.86 SKP2 (0.47) SKP2ALDH1A1CYP1A2ALOX15CASP7
SCHEMBL23093069 0.85 ALDH1A1 (0.59) SKP2ALDH1A1CYP1A2ALOX15CASP7
SCHEMBL10615570 0.82 ALDH1A1 (0.55) SKP2ALDH1A1CYP1A2ALOX15CASP7
SCHEMBL5379612 0.80 SKP2 (0.42) SKP2ALDH1A1CYP1A2ALOX15CASP7
SCHEMBL11114074 0.79 TLR8 (0.46) SKP2ALOX15CYP3A4TSHRTLR8
SCHEMBL841582 0.77 ALOX5 (0.47) ALOX15CYP3A4TSHRTLR8TYR
SCHEMBL15486053 0.77 ALOX5 (0.47) ALOX15CYP3A4TSHRTLR8TYR
SCHEMBL31265135 0.77 TYR (0.41) SKP2ALDH1A1ALOX15MAPK1CYP3A4
SCHEMBL27671383 0.77 SKP2 (0.44) SKP2ALDH1A1CYP1A2ALOX15CASP7
SCHEMBL11276129 0.77 SKP2 (0.44) SKP2ALDH1A1ALOX15MAPK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3290419-A1 FUSED-RING OR TRICYCLIC ARYL PYRIMIDINE COMPOUND USED AS KINASE INHIBITOR GUANGDONG ZHONGSHENG PHARMACEUTICAL CO., LTD (CN) 2018-03-07 EP disclosed
EP-2880026-B1 DIHYDROPYRIDONE P1 AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-02-22 EP disclosed