SCHEMBL1857795

SCHEMBL1857795

Clc1[c]c(Cl)c(Cc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTRC Q99895 3/20 0.44
CALM1 P0DP23 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
HIF1A Q16665 1/20 0.42
HSD17B10 Q99714 1/20 0.42
BCL2 P10415 1/20 0.41
BCL2L1 Q07817 1/20 0.41
ALOX5 P09917 1/20 0.40
HTR2A P28223 1/20 0.38
NR1H2 P55055 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3540407 0.84 MEN1 (0.46) MEN1KMT2ACYP3A4HPGDALOX15
SCHEMBL1862187 0.81 MAPT (0.36) MEN1KMT2AHPGDALDH1A1
SCHEMBL1859756 0.81 IDO1 (0.34) MEN1KMT2AALDH1A1
SCHEMBL1859749 0.79 TAAR1 (0.37) KMT2AHPGDALDH1A1
SCHEMBL1859772 0.77 LTA4H (0.46) HPGDALOX15ALOX5ALDH1A1
SCHEMBL1865021 0.73 SLC6A4 (0.35) HPGDHTR2A
SCHEMBL7463754 0.72 HTR2A (0.42) CTRCCALM1MEN1KMT2ACYP3A4
SCHEMBL1862207 0.72 IDO1 (0.45) MEN1KMT2AALDH1A1
SCHEMBL1046166 0.71 CALM1 (0.58) CTRCCALM1MEN1KMT2ACYP3A4
SCHEMBL1860328 0.70 CTRC (0.39) CTRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052498-A1 3,7-DIAZABICYCLO[3.3.1]NONANE CARBOXAMIDES AS ANTITHROMBOTIC AGENTS Council of Scientific & Industrial Research (IN) 2016-08-10 EP disclosed
WO-2015044951-A1 3,7-DIAZABICYCLO[3.3.1 ]NONANE CARBOXAMIDES AS ANTITHROMBOTIC AGENTS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-04-02 WO disclosed
US-7939509-B2 Partial and full agonists of A1 adenosine receptors GILEAD SCIENCES, INC. (US) 2011-05-10 US disclosed
EP-1140900-A4 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY INC (US) 2002-04-10 EP disclosed
EP-1140900-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2001-10-10 EP disclosed
WO-2000039083-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2000-07-06 WO disclosed