SCHEMBL1857797

SCHEMBL1857797

Clc1[c]c(Cl)cc(Cc2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.55
IDH1 O75874 1/20 0.42
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
BCL2 P10415 1/20 0.40
BCL2L1 Q07817 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LTA4H P09960 1/20 0.39
PTPN1 P18031 3/20 0.38
PTPN2 P17706 1/20 0.38
PTPN6 P29350 1/20 0.38
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
PLA2G10 O15496 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859758 0.78 SRD5A2 (0.39) MEN1CYP3A4KMT2AHIF1AALDH1A1
SCHEMBL1862188 0.78 IDO1 (0.38) CYP3A4KMT2A
SCHEMBL28173954 0.77 CALM1 (0.80) CALM1IDH1BCL2BCL2L1ALDH1A1
SCHEMBL7463762 0.77 CALM1 (0.48) CALM1IDH1MEN1CYP3A4HPGD
SCHEMBL16770503 0.76 CALM1 (0.60) CALM1IDH1MEN1CYP3A4HPGD
SCHEMBL27934848 0.76 CALM1 (0.60) CALM1IDH1MEN1CYP3A4HPGD
SCHEMBL1859752 0.75 TAAR1 (0.39) LTA4HLMNA
SCHEMBL2091627 0.74 CALM1 (0.57) CALM1IDH1BCL2BCL2L1LTA4H
Hydrogen Sulfide SCHEMBL28232332 0.74 CALM1 (0.57) CALM1IDH1MEN1CYP3A4HPGD
SCHEMBL1859774 0.74 LTA4H (0.55) ALOX15ALDH1A1LTA4HLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052498-A1 3,7-DIAZABICYCLO[3.3.1]NONANE CARBOXAMIDES AS ANTITHROMBOTIC AGENTS Council of Scientific & Industrial Research (IN) 2016-08-10 EP disclosed
WO-2015044951-A1 3,7-DIAZABICYCLO[3.3.1 ]NONANE CARBOXAMIDES AS ANTITHROMBOTIC AGENTS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-04-02 WO disclosed
US-7939509-B2 Partial and full agonists of A1 adenosine receptors GILEAD SCIENCES, INC. (US) 2011-05-10 US disclosed
EP-1140900-A4 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY INC (US) 2002-04-10 EP disclosed
EP-1140900-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2001-10-10 EP disclosed
WO-2000039083-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2000-07-06 WO disclosed