SCHEMBL1859758

SCHEMBL1859758

Cc1ccc(Cc2cc(Cl)[c]c(Cl)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.39
IDO1 P14902 1/20 0.38
CYP3A4 P08684 2/20 0.37
DAO P14920 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
KMT2A Q03164 2/20 0.36
ALOX12 P18054 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35
LTA4H P09960 1/20 0.35
AGXT P21549 2/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1862188 0.79 IDO1 (0.38) IDO1CYP3A4DAOCYP2C19KMT2A
SCHEMBL1859774 0.79 LTA4H (0.55) IDO1KDM4ECYP2C19CYP1A2TAAR1
SCHEMBL1857797 0.78 CALM1 (0.55) CYP3A4HIF1AKMT2ALTA4HMEN1
SCHEMBL1149394 0.76 IDO1 (0.58) SRD5A2IDO1CYP3A4DAOKMT2A
SCHEMBL11410252 0.76 IDO1 (0.58) SRD5A2IDO1CYP3A4DAOKMT2A
SCHEMBL11844782 0.75 IDO1 (0.46) SRD5A2IDO1CYP3A4DAOCYP1A2
SCHEMBL10389845 0.75 RAB9A (0.53) SRD5A2IDO1KMT2AALOX12TAAR1
SCHEMBL14270799 0.73 CYP3A4 (0.42) SRD5A2CYP3A4CYP2C19KMT2ACYP1A2
SCHEMBL1859752 0.72 TAAR1 (0.39) KDM4ETAAR1LTA4HMAPTNPC1
SCHEMBL14397402 0.71 CYP3A4 (0.47) SRD5A2IDO1CYP3A4DAOKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7939509-B2 Partial and full agonists of A1 adenosine receptors GILEAD SCIENCES, INC. (US) 2011-05-10 US disclosed