SCHEMBL1859752

SCHEMBL1859752

Cc1ccccc1Cc1cc(Cl)[c]c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
TYMP P19971 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LTA4H P09960 1/20 0.36
KDR P35968 1/20 0.35
AR P10275 1/20 0.35
POLB P06746 1/20 0.35
CHRM2 P08172 1/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
MAPT P10636 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1862185 0.79 CYP1A2 (0.41) TAAR1MAPT
SCHEMBL1862209 0.79 IDO1 (0.46) TAAR1SLC6A2SLC6A4SLC6A3LTA4H
SCHEMBL1861221 0.77 KDM4E (0.44) LTA4HARPOLBKDM4E
SCHEMBL1857797 0.75 CALM1 (0.55) LTA4HLMNA
SCHEMBL1859749 0.74 TAAR1 (0.37) TAAR1TYMPNPC1RAB9ALTA4H
SCHEMBL8095627 0.74 LTA4H (0.53) TAAR1SLC6A2SLC6A4SLC6A3LTA4H
SCHEMBL11303064 0.74 MAPK1 (0.47) TAAR1SLC6A2SLC6A4SLC6A3NPC1
SCHEMBL29477327 0.73 TAAR1 (0.56) TAAR1TYMPLTA4HARCHRM2
SCHEMBL2090458 0.73 TAAR1 (0.56) TAAR1TYMPLTA4HARCHRM2
SCHEMBL1859758 0.72 SRD5A2 (0.39) TAAR1NPC1RAB9ALTA4HMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7939509-B2 Partial and full agonists of A1 adenosine receptors GILEAD SCIENCES, INC. (US) 2011-05-10 US disclosed