SCHEMBL18600014

SCHEMBL18600014

INc1cnc2ccccc2c1N1CCNCC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 4/20 0.50
ADRB2 P07550 2/20 0.50
PDE10A Q9Y233 1/20 0.44
BCHE P06276 6/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
KDM1A O60341 1/20 0.41
ADRB1 P08588 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
GRM5 P41594 2/20 0.40
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13322696 0.86 NCF1 (0.50) NCF1ADRB2PDE10ABCHECHRNB2
SCHEMBL13354913 0.78 NCF1 (0.54) NCF1ADRB2PDE10ACHRNB2CHRNA4
SCHEMBL29974103 0.75 ADRB2 (0.50) NCF1ADRB2PDE10AHPGD
SCHEMBL25292523 0.75 MAOB (0.46) NCF1ADRB2PDE10ABCHE
SCHEMBL31145260 0.75 MAOB (0.46) NCF1ADRB2PDE10ABCHE
SCHEMBL21781663 0.69 GRM5 (0.54) BCHEGRM5
SCHEMBL31423816 0.68 NCF1 (0.51) NCF1ADRB2CHRNB2CHRNA4ADRB1
SCHEMBL900231 0.67 NCF1 (1.00) NCF1ADRB2ADRB1ALDH1A1HPGD
SCHEMBL29936658 0.67 PTK2 (0.67) NCF1ADRB2ALDH1A1HPGDHTR2C
SCHEMBL30041391 0.67 NCF1 (1.00) NCF1ADRB2ADRB1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078003-B1 ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF MERCK SHARP & DOHME (US) 2017-03-08 EP disclosed