SCHEMBL18600545

SCHEMBL18600545

CCN(Cc1ccc(F)cc1)c1ccc(N=C=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.47
CNR1 P21554 5/20 0.47
TSHR P16473 2/20 0.46
CYP3A4 P08684 1/20 0.46
LMNA P02545 1/20 0.46
GRIA2 P42262 6/20 0.43
GRIN2A Q12879 5/20 0.43
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18600540 0.83 KCNQ4 (0.48) CNR2CNR1TSHRCYP3A4
SCHEMBL2853713 0.82 ALDH1A1 (0.53) CNR2TSHRCYP3A4LMNAALDH1A1
SCHEMBL5909497 0.81 CYP3A4 (0.67) CNR2CNR1TSHRCYP3A4LMNA
SCHEMBL27689884 0.76 TSHR (0.75) CNR2CNR1TSHRLMNAGRIA2
SCHEMBL93163 0.75 CYP3A4 (0.56) TSHRCYP3A4ALDH1A1MAPTMAPK1
SCHEMBL22340467 0.74 CNR2 (0.51) CNR2CNR1TSHRLMNAALDH1A1
Ether SCHEMBL596696 0.73 CYP3A4 (0.47) TSHRCYP3A4LMNAALDH1A1KDM4E
SCHEMBL12069745 0.72 MAPT (0.54) CNR2CNR1TSHRCYP3A4LMNA
SCHEMBL6984098 0.71 ALDH1A1 (0.66) CNR2CNR1TSHRCYP3A4LMNA
SCHEMBL18600203 0.70 PYCR1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138833-A1 NOVEL KCNQ POTASSIUM CHANNEL AGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2017-03-08 EP disclosed