SCHEMBL1862897

SCHEMBL1862897

c1ccc(C2(c3cccnc3)CCCC[N]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
P2RX7 Q99572 1/20 0.37
OPRM1 P35372 2/20 0.37
OPRL1 P41146 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
VNN1 O95497 1/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
CNR2 P34972 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
HCAR2 Q8TDS4 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1862411 0.95 ALDH1A1 (0.40) LMNAALDH1A1P2RX7OPRM1OPRL1
SCHEMBL1866642 0.95 ALDH1A1 (0.40) LMNAALDH1A1P2RX7OPRM1OPRL1
SCHEMBL1865507 0.90 ALDH1A1 (0.42) LMNAALDH1A1OPRM1OPRL1MEN1
SCHEMBL9639574 0.86 DPP4 (0.41) LMNAOPRM1NPSR1OPRD1
SCHEMBL1863575 0.79 CHRNB2 (0.37) LMNAALDH1A1MEN1KMT2ACYP3A4
SCHEMBL5760516 0.77 SLC6A3 (0.39) S1PR1
SCHEMBL1866073 0.75 HTR2A (0.38) LMNAALDH1A1OPRM1OPRL1MEN1
SCHEMBL1865938 0.75 HTR2A (0.38) LMNAALDH1A1OPRM1OPRL1MEN1
SCHEMBL1860147 0.75 HTR2A (0.38) LMNAALDH1A1OPRM1OPRL1MEN1
SCHEMBL23722370 0.68 ALDH1A1 (0.55) LMNAALDH1A1OPRM1OPRL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493877-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS Janssen Pharmaceutica NV (BE) 2012-09-05 EP disclosed
WO-2011053705-A1 PYRIMIDINE COMPOUNDS AS DELTA OPIOID RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-05-05 WO disclosed