SCHEMBL1863285

SCHEMBL1863285

CN(C[C@@H](N)[C@@H](O)C1CCCCC1)C(=O)OCC[Si](C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
METAP2 P50579 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1859646 1.00 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3CHRNB2CHRNB4
SCHEMBL1860870 0.99 CHRNB2 (0.33) SLC6A2SLC6A4SLC6A3CHRNB2CHRNB4
SCHEMBL970253 0.81 REN (0.40) METAP2
SCHEMBL3607292 0.79 CTSK (0.36) METAP2
SCHEMBL3607293 0.79 CTSK (0.36) METAP2
SCHEMBL499255 0.79 CTSK (0.36) METAP2
SCHEMBL499254 0.79 CTSK (0.36) METAP2
SCHEMBL1866972 0.79 L3MBTL1 (0.31) SLC6A2SLC6A4SLC6A3L3MBTL1
SCHEMBL1863059 0.79 L3MBTL1 (0.31) SLC6A2SLC6A4SLC6A3L3MBTL1
SCHEMBL1866462 0.78 CTSK (0.34) CHRNB2CHRNB4CHRNA3CHRNA4METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. 2011-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors DNPEP, PEPD, ACE SLC6A2 3389/4885SLC6A4 3809/4885SLC6A3 2752/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.