SCHEMBL18654366

SCHEMBL18654366

Cc1cc(N)cc(OCCCOC(C)(C)O)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 2/20 0.44
KMT2A Q03164 2/20 0.37
THRB P10828 1/20 0.37
POLB P06746 2/20 0.35
LTB4R Q15722 2/20 0.33
KCNH2 Q12809 1/20 0.33
ALDH1A1 P00352 3/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP2C19 P33261 2/20 0.32
MEN1 O00255 1/20 0.32
GLA P06280 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2457239 0.77 ALDH1A1 (0.49) NUDT1KMT2ATHRBPOLBKCNH2
SCHEMBL22239676 0.74 ALOX5AP (0.36) NUDT1
SCHEMBL17778688 0.74 KDM4E (0.44) KMT2APOLBLTB4RALDH1A1MAPT
SCHEMBL22119490 0.73 NUDT1 (0.41) NUDT1KMT2ATHRBPOLBKCNH2
SCHEMBL18654717 0.73 MCHR1 (0.37) NUDT1
SCHEMBL18654540 0.73 CDK2 (0.31) NUDT1KMT2AMAPTMEN1
SCHEMBL17778782 0.72 FEN1 (0.32)
SCHEMBL17778488 0.71 KDM4E (0.35)
SCHEMBL20606933 0.71 SMN1; SMN2 (0.45) NUDT1KMT2APOLBALDH1A1LMNA
SCHEMBL22239544 0.70 CHRNB2 (0.35) TSHRAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2768509-B1 SUBSTITUTED BICYCLIC AZA-HETEROCYCLES AND ANALOGUES AS SIRTUIN MODULATORS GLAXOSMITHKLINE LLC (US) 2017-03-22 EP disclosed