SCHEMBL1871663

SCHEMBL1871663

CCCn1c(NCc2ccccc2OC)nc(=O)c2c1N=C(C1CCCC1)[N]2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.45
MAPT P10636 2/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
TSHR P16473 2/20 0.44
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 3/20 0.44
GAA P10253 2/20 0.44
PKM P14618 2/20 0.44
P2RX7 Q99572 2/20 0.43
LMNA P02545 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HTT P42858 2/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
PDE9A O76083 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.39
F2 P00734 1/20 0.39
MAPK1 P28482 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1871541 0.81 HTT (0.44) SMN1; SMN2TSHRALDH1A1GAALMNA
SCHEMBL1872803 0.79 ADORA1 (0.59) MAPTGAAP2RX7PDE9AADORA1
SCHEMBL1868348 0.78 ADORA1 (0.58) TP53MAPTGAAP2RX7PDE9A
SCHEMBL1866236 0.78 ADORA1 (0.41) MAPTTSHRALDH1A1MEN1KMT2A
SCHEMBL1873285 0.74 ADORA1 (0.69) ADORA1
SCHEMBL1875802 0.74 ADORA1 (0.44) ALDH1A1GAAKDM4EADORA1
SCHEMBL1868690 0.74 ADORA1 (0.57) ADORA1
SCHEMBL1870248 0.73 ADORA3 (0.39) PKMKMT2AADORA1
SCHEMBL1887812 0.73 ADORA2B (0.39) TSHRLMNAMEN1KMT2AADORA1
SCHEMBL1871164 0.72 ADORA1 (0.45) TP53HTTADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499142-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF Advinus Therapeutics Limited (IN) 2012-09-19 EP disclosed
WO-2011055391-A1 SUBSTITUTED FUSED PYRIMIDINE COMPOUNDS, ITS PREPARATION AND USES THEREOF ADVINUS THERAPEUTICS PRIVATE LIMITED (IN) 2011-05-12 WO disclosed