SCHEMBL18790992

SCHEMBL18790992

Cc1ccccc1-c1cncc(N2CCNCC2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.60
CYP3A4 P08684 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP2D6 P10635 2/20 0.53
TSHR P16473 2/20 0.53
RECQL P46063 1/20 0.53
HTR7 P34969 2/20 0.52
HTR1A P08908 2/20 0.50
HTR2A P28223 2/20 0.50
HTR2C P28335 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CLK4 Q9HAZ1 1/20 0.48
PIM2 Q9P1W9 7/20 0.47
PIM1 P11309 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29161357 0.83 HTR2C (0.50) CYP1A2CYP3A4MEN1KMT2AHTR7
SCHEMBL4997526 0.83 CYP11B2 (0.51) CYP1A2TSHRKDM4EALDH1A1HPGD
SCHEMBL5003463 0.81 CYP11B2 (0.49) CYP1A2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL3530819 0.80 PIM2 (0.48) CYP1A2CYP3A4MEN1KMT2AHTR7
SCHEMBL4992085 0.79 MAPT (0.52) CYP1A2KMT2AKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL3269195 0.78 PIM2 (0.61) CYP1A2CYP3A4MEN1KMT2AHTR7
SCHEMBL22236781 0.77 ROCK2 (0.58) CYP1A2CYP3A4MEN1KMT2AHTR7
SCHEMBL5000713 0.77 LMNA (0.57) CYP1A2CYP3A4MEN1KMT2ATSHR
SCHEMBL18502904 0.77 CYP11B2 (0.66) CYP1A2CYP3A4MEN1KMT2ACYP2D6
SCHEMBL5002999 0.76 DHFR (0.45) MEN1KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3381904-B1 NOVEL NITROGEN-CONTAINING AROMATIC HETEROCYCLIC COMPOUND MITSUBISHI TANABE PHARMA CORP (JP) 2021-07-28 EP disclosed
US-10717731-B2 Nitrogen-containing aromatic heterocyclic compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2020-07-21 US disclosed
WO-2017069226-A1 NOVEL NITROGEN-CONTAINING AROMATIC HETEROCYCLIC COMPOUND 田辺三菱製薬株式会社 2017-04-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10717731-B2 Nitrogen-containing aromatic heterocyclic compound REN, NR3C2, NR5A1 CYP1A2 645/4885CYP3A4 2134/4885MEN1 734/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.