SCHEMBL18794837

SCHEMBL18794837

O=C1NCCCCC1(F)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.38
OPRM1 P35372 2/20 0.38
KCNH2 Q12809 1/20 0.38
SLC6A3 Q01959 3/20 0.38
HSD11B1 P28845 1/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2A Q12879 2/20 0.37
POLB P06746 1/20 0.36
DAO P14920 1/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18822478 0.85 DRD2 (0.38) SLC6A9OPRM1SLC6A3HSD11B1GRIN1
SCHEMBL18794831 0.85 DRD2 (0.38) SLC6A9OPRM1SLC6A3HSD11B1GRIN1
SCHEMBL18822477 0.85 DRD2 (0.38) SLC6A9OPRM1SLC6A3HSD11B1GRIN1
SCHEMBL18794819 0.85 GRIN1 (0.51) SLC6A9OPRM1GRIN1GRIN2APOLB
SCHEMBL18794833 0.83 METAP2 (0.38) GRIN1GRIN2AGRIN2B
SCHEMBL28546096 0.80 GRIN1 (0.43) GRIN1GRIN2AGRIN2BMAOAMAOB
SCHEMBL18794865 0.79 SLC6A3 (0.46) SLC6A3GRIN1GRIN2ASLC6A4SLC6A2
SCHEMBL18794835 0.79 HSD11B1 (0.40) SLC6A9OPRM1KCNH2SLC6A3HSD11B1
SCHEMBL18794816 0.78 SLC6A4 (0.42) KCNH2SLC6A3SLC6A4SLC6A2
SCHEMBL18794813 0.77 METAP2 (0.41) GRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017070793-A1 NOVEL FLUORINATED HETEROCYCLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS TRILLIUM THERAPEUTICS INC. (CA) 2017-05-04 WO claimed
WO-2017070793-A1 NOVEL FLUORINATED HETEROCYCLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS TRILLIUM THERAPEUTICS INC. (CA) 2017-05-04 WO disclosed
WO-2017070793-A1 NOVEL FLUORINATED HETEROCYCLE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS TRILLIUM THERAPEUTICS INC. (CA) 2017-05-04 WO disclosed