SCHEMBL18828601

SCHEMBL18828601

CN1CCN([S+]([O-])c2ccc(Br)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
DUSP3 P51452 2/20 0.44
PTPN5 P54829 2/20 0.44
PTPN11 Q06124 2/20 0.44
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 3/20 0.39
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
KDM4E B2RXH2 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
HRH4 Q9H3N8 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22340249 0.82 HPGD (0.37) ALDH1A1RAB9ANPC1LMNAPOLB
SCHEMBL14547446 0.81 MAPT (0.48) ALDH1A1LMNAPOLBMAPTKDM4E
SCHEMBL22643223 0.81 HPGD (0.36) ALDH1A1RAB9ANPC1LMNAPOLB
SCHEMBL6595771 0.81 DUSP3 (0.49) ALDH1A1DUSP3PTPN5PTPN11MAPT
SCHEMBL1370673 0.78 HPGD (0.35) MAPTMAPK1HTR1DHTR1BHTR2A
SCHEMBL18828660 0.77 CA2 (0.35)
SCHEMBL3773093 0.76 DPP4 (0.34)
SCHEMBL20310914 0.74 KDM4E (0.34) KDM4ESMN1; SMN2
SCHEMBL24181233 0.73 RAB9A (0.42) ALDH1A1DUSP3PTPN5PTPN11RAB9A
SCHEMBL21613823 0.72 DHCR7 (0.39) RAB9APOLBKDM4EHRH3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970228-B1 SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2017-05-10 EP disclosed