SCHEMBL188333

SCHEMBL188333

C=CC(=O)Oc1cc(F)cc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.42
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
CES2 O00748 2/20 0.39
CES1 P23141 2/20 0.39
TGM2 P21980 1/20 0.34
TP53 P04637 4/20 0.33
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
CYP3A4 P08684 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
EGFR P00533 1/20 0.33
PKM P14618 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
JAK1 P23458 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11850804 0.84 THRB (0.48) THRBTGM2TP53ALDH1A1MAPT
SCHEMBL2604617 0.82 THRB (0.44) THRBCYP4F2CYP4A11TP53MAPT
SCHEMBL10181369 0.81 CES2 (0.41) THRBCYP4F2CYP4A11CES2CES1
SCHEMBL1098081 0.81 THRB (0.41) THRBCYP4F2CYP4A11TP53ALDH1A1
SCHEMBL30543222 0.80 ESR1 (0.49) THRBCES2CES1ALDH1A1MEN1
SCHEMBL5634217 0.80 ESR1 (0.49) THRBCES2CES1ALDH1A1MEN1
SCHEMBL27495352 0.80 CYP4F2 (0.43) CYP4F2CYP4A11CES2CES1TP53
SCHEMBL10179885 0.79 ERN1 (0.38) THRBCES2CES1TGM2MAPK1
SCHEMBL2604634 0.79 HSD17B1 (0.39) THRBMAPTCYP3A4MEN1KMT2A
SCHEMBL2975869 0.78 THRB (0.55) THRBCES2CES1TGM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2400844-A1 STEREOSELECTIVE HYDROGENATION OF A KETONE Glaxo Group Limited (GB) 2012-01-04 EP claimed
WO-2010099098-A1 STEREOSELECTIVE HYDROGENATION OF A KETONE GLAXO GROUP LIMITED (GB) 2010-09-02 WO claimed
CN-112679495-B Estrogen receptor modulators 里科瑞尔姆IP控股有限责任公司 2023-03-28 CN disclosed
CN-104112870-A Nonaqueous electrolyte solution and nonaqueous electrolyte battery using same MITSUBISHI CHEM CORP 2014-10-22 CN disclosed
US-20130244122-A1 NONAQUEOUS ELECTROLYTIC SOLUTION AND NONAQUEOUS-ELECTROLYTE BATTERY EMPLOYING THE SAME ONUKI MASAMICHI (JP) 2013-09-19 US disclosed
US-20120219866-A1 NONAQUEOUS ELECTROLYTIC SOLUTION AND NONAQUEOUS-ELECTROLYTE BATTERY EMPLOYING THE SAME MITSUBISHI CHEMICAL CORPORATION (JP) 2012-08-30 US disclosed
EP-2475041-A1 NON-AQUEOUS ELECTROLYTIC SOLUTION, AND NON-AQUEOUS ELECTROLYTE BATTERY COMPRISING SAME Mitsubishi Chemical Corporation (JP) 2012-07-11 EP disclosed
CN-102484281-A Nonaqueous electrolyte solution and nonaqueous electrolyte battery using same MITSUBISHI CHEM CORP 2012-05-30 CN disclosed