SCHEMBL18862275

SCHEMBL18862275

CCOC(=O)C1CCCN(Cc2ccc(-c3ccccc3[N+](=O)[O-])o2)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
PKM P14618 1/20 0.59
CYP2C19 P33261 1/20 0.59
KMT2A Q03164 2/20 0.56
ALDH1A1 P00352 8/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
IL33 O95760 2/20 0.53
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MAPK1 P28482 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
MAPT P10636 3/20 0.52
TDP1 Q9NUW8 1/20 0.52
MEN1 O00255 1/20 0.51
USP2 O75604 1/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18862272 0.82 IL33 (0.55) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL18862278 0.77 MAPT (0.59) KDM4ECYP1A2CYP3A4CYP2C9PKM
SCHEMBL18862279 0.74 IL33 (0.52) KDM4EPKMKMT2AALDH1A1SMN1; SMN2
SCHEMBL3435049 0.74 ALDH1A1 (0.70) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28972131 0.73 ALDH1A1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28972130 0.73 ALDH1A1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31687195 0.73 ALDH1A1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1946258 0.73 L3MBTL1 (0.86) KDM4EALDH1A1SMN1; SMN2ATML3MBTL1
Bromide SCHEMBL10462008 0.72 L3MBTL1 (0.84) KDM4EALDH1A1SMN1; SMN2ATML3MBTL1
SCHEMBL18862291 0.69 IL33 (1.00) KDM4EPKMKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017083242-A1 INHIBITORS OF SUPPRESSION OF TUMORIGENCITY 2 (ST2) AND METHODS USING THE SAME THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2017-05-18 WO disclosed