SCHEMBL18895992

SCHEMBL18895992

COc1ccc2c(c1)C(CCCN1CCC(N)(c3ccccc3)CC1)c1cccnc1CO2

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.40
HTR1A P08908 2/20 0.36
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 1/20 0.35
HTR7 P34969 1/20 0.34
HSPA9 P38646 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2B P41595 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7615965 0.78 HTR1A (0.35) SIGMAR1HTR1AMEN1ALDH1A1KMT2A
SCHEMBL10287635 0.71 CCR1 (0.49) HTR1AALDH1A1HRH3DRD2DRD3
SCHEMBL10702160 0.70 HTR2B (0.40) SIGMAR1HTR1AMEN1ALDH1A1LMNA
SCHEMBL10699642 0.69 EDNRB (0.41) SIGMAR1HTR1AMEN1ALDH1A1KMT2A
SCHEMBL12121748 0.68 CCR1 (0.37) DRD2DRD3DRD4
SCHEMBL8800043 0.68 DRD2 (0.36) SIGMAR1HTR1AMEN1ALDH1A1KMT2A
SCHEMBL10287667 0.68 CCR1 (0.54) SIGMAR1MEN1ALDH1A1LMNAKMT2A
SCHEMBL8797672 0.67 EDNRB (0.46) MEN1ALDH1A1KMT2ADRD2DRD3
SCHEMBL7205528 0.67 CCR1 (0.49) KMT2AOPRM1OPRD1
SCHEMBL7205522 0.67 CCR1 (0.49) KMT2AOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663537-B2 Chemokine receptor antagonists and methods of use MILLENNIUM PHARMACEUTICALS, INC. (US) 2017-05-30 US disclosed