SCHEMBL7615965

SCHEMBL7615965

COc1ccc2c(c1)C(CCCBr)c1cccnc1CO2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.35
HTR2B P41595 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
HTR2A P28223 4/20 0.35
ALDH1A1 P00352 4/20 0.35
MAPT P10636 3/20 0.35
GAA P10253 2/20 0.35
HPGD P15428 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALOX12 P18054 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
P2RX7 Q99572 1/20 0.34
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10699642 0.79 EDNRB (0.41) HTR1AHTR2BSIGMAR1HTR2AALDH1A1
SCHEMBL10702160 0.78 HTR2B (0.40) HTR1AHTR2BSIGMAR1HTR2AALDH1A1
SCHEMBL18895992 0.78 SIGMAR1 (0.40) HTR1AHTR2BSIGMAR1ALDH1A1DRD2
SCHEMBL8800043 0.76 DRD2 (0.36) HTR1AHTR2BSIGMAR1ALDH1A1MAPT
SCHEMBL7209964 0.75 EDNRB (0.36) HTR1AHTR2BSIGMAR1ALDH1A1MAPT
SCHEMBL8797672 0.75 EDNRB (0.46) ALDH1A1MAPTGAAHPGDTDP1
SCHEMBL2215953 0.70 HTR2A (0.55) HTR1AHTR2BSIGMAR1HTR2AALDH1A1
SCHEMBL2217095 0.70 HTR2A (0.55) HTR2AALDH1A1MAPTGAAHPGD
SCHEMBL7210858 0.70 ALDH1A1 (0.42) HTR1AHTR2BSIGMAR1HTR2AALDH1A1
SCHEMBL7210855 0.70 ALDH1A1 (0.42) HTR1AHTR2BSIGMAR1HTR2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6433165-B1 ANTIINFLAMMATORY AGENTS MILLENNIUM PHARMACEUTICALS, INC. 2002-08-13 US disclosed