SCHEMBL18901313

SCHEMBL18901313

Cc1ccc2c(c1)[nH]c1cncc(F)c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.49
ROCK2 O75116 5/20 0.48
GABRA1 P14867 3/20 0.48
GABRG2 P18507 3/20 0.48
GABRB3 P28472 3/20 0.48
GABRA5 P31644 3/20 0.48
GABRA3 P34903 3/20 0.48
GABRA2 P47869 3/20 0.48
GABRP O00591 2/20 0.48
GABRD O14764 2/20 0.48
GABRB1 P18505 2/20 0.48
GABRB2 P47870 2/20 0.48
GABRA4 P48169 2/20 0.48
GABRE P78334 2/20 0.48
GABRA6 Q16445 2/20 0.48
GABRG1 Q8N1C3 2/20 0.48
GABRG3 Q99928 2/20 0.48
GABRQ Q9UN88 2/20 0.48
ACHE P22303 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18901227 0.83 GABRP (0.50) KIF11ROCK2GABRA1GABRG2GABRB3
SCHEMBL28050860 0.77 KIF11 (0.56) KIF11GABRA1GABRG2GABRB3GABRA5
SCHEMBL16345630 0.76 ROCK2 (0.62) KIF11ROCK2
SCHEMBL2628365 0.73 ACHE (0.59) KIF11GABRA1GABRG2GABRB3GABRA5
SCHEMBL4256780 0.72 KIF11 (0.78) KIF11GABRA1GABRG2GABRB3GABRA5
SCHEMBL29518339 0.72 KIF11 (0.78) KIF11GABRA1GABRG2GABRB3GABRA5
SCHEMBL1798677 0.71 CHUK (0.55) ROCK2GABRA1GABRG2GABRB3GABRA5
SCHEMBL23369904 0.70 KIF11 (0.82) KIF11ACHERXFP1
SCHEMBL18901304 0.69 KIF11 (0.58) KIF11ROCK2GABRA1GABRG2GABRB3
SCHEMBL2628321 0.69 GABRP (0.49) KIF11GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016951-B1 TRICYCLIC PYRIDO-CARBOXAMIDE DERIVATIVES AS ROCK INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed