SCHEMBL18909248

SCHEMBL18909248

CCC(=O)N1CCC(N2CCC(C#N)C2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 1/20 0.42
CHRM1 P11229 2/20 0.40
EPHX2 P34913 4/20 0.39
CHRM2 P08172 1/20 0.38
ALDH1A1 P00352 1/20 0.37
EPHX1 P07099 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA3 P32297 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB3 Q05901 1/20 0.36
CHRNA6 Q15825 1/20 0.36
PKM P14618 1/20 0.35
KDM6B O15054 1/20 0.35
KDM5C P41229 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM2A Q9Y2K7 1/20 0.35
KDM3A Q9Y4C1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18909103 0.92 PKM (0.41) KDM2BCHRM1EPHX2ALDH1A1PKM
SCHEMBL22891320 0.92 PKM (0.41) KDM2BCHRM1EPHX2ALDH1A1PKM
SCHEMBL21281054 0.92 PKM (0.41) KDM2BCHRM1EPHX2ALDH1A1PKM
SCHEMBL23514580 0.91 CHRM1 (0.44) KDM2BCHRM1EPHX2CHRM2ALDH1A1
SCHEMBL22891271 0.85 DPP4 (0.42) KDM2BCHRM1
SCHEMBL16621798 0.84 CHRNB2 (0.42) EPHX2ALDH1A1EPHX1JAK2JAK1
SCHEMBL13045920 0.84 EPHX2 (0.47) EPHX2ALDH1A1EPHX1CHRNB2CHRNA3
SCHEMBL24585220 0.79 MGLL (0.39) KDM2BCHRM1EPHX2ALDH1A1KDM4E
SCHEMBL24585219 0.79 MGLL (0.39) KDM2BCHRM1EPHX2ALDH1A1KDM4E
SCHEMBL24521475 0.77 SMN1; SMN2 (0.43) CHRM1EPHX2CHRM2ALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017089390-A1 JANUS KINASES INHIBITORS, COMPOSITIONS THEREOF AND USE THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-06-01 WO disclosed