SCHEMBL1892146

SCHEMBL1892146

O=S(=O)(O)OCC(COS(=O)(=O)O)COS(=O)(=O)O

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.37
CA1 P00915 2/20 0.36
CA12 O43570 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718720 0.86 CA2 (0.32) CA2CA1CA12CA7CA14
SCHEMBL15215211 0.84 CA2 (0.40) CA2CA1CA12CA7CA14
SCHEMBL1425858 0.79 CA2 (0.35) CA2TSHRTDP1
SCHEMBL15773891 0.79
SCHEMBL13997140 0.77
SCHEMBL13254849 0.77
SCHEMBL25235825 0.77
SCHEMBL9651396 0.77 CA2 (0.56) CA2CA1TSHRTDP1CA9
SCHEMBL4667979 0.77
SCHEMBL8329628 0.77 CA2 (0.33) CA2CA1CA7TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064013-A4 $i(IN VITRO) FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIV WASHINGTON (US) 2005-05-11 EP claimed
EP-1064013-A1 $i(IN VITRO) FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES University of Washington (US) 2001-01-03 EP claimed
WO-1999045947-A9 IN VITRO FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIV WASHINGTON (US) 2000-03-02 WO claimed
WO-1999045947-A1 IN VITRO FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIVERSITY OF WASHINGTON (US) 1999-09-16 WO claimed
US-20140155480-A1 Scyllo-Inositol Derivatives and Their Use in the Treatment of Diseases Characterized by Abnormal Protein Folding or Aggregation of Amyloid Formation, Deposition, Accumulation for Persistence WARATAH PHARMACEUTICALS INC. (CA) 2014-06-05 US disclosed
US-20140135403-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF OCULAR DISEASES WARATAH PHARMACEUTICALS INC. (CA) 2014-05-15 US disclosed
EP-2656839-A1 Use of Cyclohexanehexol Derivatives in the Treatment of Ocular Diseases Waratah Pharmaceuticals, Inc. (CA) 2013-10-30 EP disclosed
US-20110105626-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES FOR THE TREATMENT OF POLYGLUTAMINE DISEASES MCLAURIN JOANNE 2011-05-05 US disclosed
US-20100331267-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF ALPHA-SYNUCLEINOPATHIES MCLAURIN JOANNE 2010-12-30 US disclosed
US-20100292157-A1 Combination Treatments for Alzheimer's Disease and Similar Diseases WARATAH PHARMACEUTICALS INC. (CA) 2010-11-18 US disclosed
US-20100173960-A1 The Combination of a Cyclohexanehexol and a NSAID for the Treatment of Neurodegenerative Diseases WARATAH PHARMACEUTICALS INC. (CA) 2010-07-08 US disclosed
US-20100168250-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF OCULAR DISEASE WARATAH PHARMACEUTICALS INC. (CA) 2010-07-01 US disclosed
US-7148001-B2 In vitro formation of congophilic maltese-cross amyloid plaques to identify anti-plaque therapeutics for the treatment of Alzheimer's and Prion diseases UNIVERSITY OF WASHINGTON (US) 2006-12-12 US disclosed
EP-1064013-A4 $i(IN VITRO) FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIV WASHINGTON (US) 2005-05-11 EP disclosed
US-20020168753-A1 In vitro formation of congophilic maltese-cross amyloid plaques to identify anti-plaque therapeutics for the treatment of Alzheimer's and Prion diseases NATIONAL INSTITUTES OF HEALTH 2002-11-14 US disclosed
EP-1064013-A1 $i(IN VITRO) FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES University of Washington (US) 2001-01-03 EP disclosed
EP-1054664-A1 METHOD FOR MODULATING MACROPHAGE ACTIVATION Neurochem, Inc. (CA) 2000-11-29 EP disclosed
WO-1999045947-A9 IN VITRO FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIV WASHINGTON (US) 2000-03-02 WO disclosed
WO-1999045947-A1 IN VITRO FORMATION OF CONGOPHILIC MALTESE-CROSS AMYLOID PLAQUES TO IDENTIFY ANTI-PLAQUE THERAPEUTICS FOR THE TREATMENT OF ALZHEIMER'S AND PRION DISEASES UNIVERSITY OF WASHINGTON (US) 1999-09-16 WO disclosed
WO-1999040909-A1 METHOD FOR MODULATING MACROPHAGE ACTIVATION NEUROCHEM, INC. (CA) 1999-08-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331267-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF ALPHA-SYNUCLEINOPATHIES SNCA, PARK7, PMP22 CA2 2600/4885CA1 2680/4885CA12 3894/4885
US-20110105626-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES FOR THE TREATMENT OF POLYGLUTAMINE DISEASES CDR2, HYPK, HTT CA2 4000/4885CA1 4311/4885CA12 4729/4885
US-20100168250-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF OCULAR DISEASE APP, IAPP, TTR CA2 1036/4885CA1 1492/4885CA12 1079/4885
US-20100292157-A1 Combination Treatments for Alzheimer's Disease and Similar Diseases APP, PSEN1, BACE1 CA2 1837/4885CA1 699/4885CA12 2973/4885
US-20100173960-A1 The Combination of a Cyclohexanehexol and a NSAID for the Treatment of Neurodegenerative Diseases HTT, APP, PSEN2 CA2 1438/4885CA1 1175/4885CA12 3183/4885
US-20140135403-A1 USE OF CYCLOHEXANEHEXOL DERIVATIVES IN THE TREATMENT OF OCULAR DISEASES APP, IAPP, TTR CA2 1094/4885CA1 1602/4885CA12 1107/4885
US-20140155480-A1 Scyllo-Inositol Derivatives and Their Use in the Treatment of Diseases Characterized by Abnormal Protein Folding or Aggregation of Amyloid Formation, Deposition, Accumulation for Persistence SCLY, SCO2, SGMS2 CA2 2349/4885CA1 3722/4885CA12 4254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.