SCHEMBL18924303

SCHEMBL18924303

CCCc1ccnc(CC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
LNPEP Q9UIQ6 5/20 0.40
NOS2 P35228 2/20 0.36
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
SREBF2 Q12772 5/20 0.35
LOX P28300 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10223946 0.88 ESR1 (0.40) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL18924478 0.87 KDM4E (0.50) KDM4ELMNACYP3A4TSHRNOS2
SCHEMBL11926806 0.85 NOS3 (0.52) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL487201 0.82 KDM4E (0.56) KDM4ELMNACYP3A4TSHRNOS2
SCHEMBL2619306 0.80 CYP1A2 (0.47) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL21533986 0.80 NOS3 (0.35) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL12561686 0.79 RECQL (0.50) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL21157383 0.79 FDPS (0.35) CYP3A4LNPEPNOS2NOS3NOS1
SCHEMBL18924506 0.79 LNPEP (0.44) KDM4ELMNACYP3A4TSHRLNPEP
SCHEMBL26433336 0.77 GRN (0.41) LMNALNPEPNOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9670172-B2 Heterocyclic compounds and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2017-06-06 US disclosed