SCHEMBL189771

SCHEMBL189771

Clc1ccc(Cl)c(CBr)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.48
CYP3A4 P08684 4/20 0.43
IDO1 P14902 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
HIF1A Q16665 2/20 0.43
SLC22A1 O15245 1/20 0.43
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43
HSP90AA1 P07900 1/20 0.43
MAPT P10636 1/20 0.43
HSPD1 P10809 1/20 0.43
HSPA5 P11021 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
CASP1 P29466 1/20 0.43
HTT P42858 1/20 0.43
BLM P54132 1/20 0.43
HSPE1 P61604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL384040 0.82 IDO1 (0.44) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL30089455 0.82 IDO1 (0.44) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL3620010 0.81 TP53 (0.44) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL1137783 0.80 IDO1 (0.60) TP53CYP3A4IDO1LMNAHTT
SCHEMBL5293792 0.78 NOS3 (0.42) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL29680819 0.78 SLC6A4 (0.39) MEN1KMT2ALMNAHPGDSMN1; SMN2
SCHEMBL30853201 0.78 MEN1 (0.41) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL532613 0.78 NOS3 (0.42) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL269490 0.78 MEN1 (0.41) TP53CYP3A4IDO1MEN1KMT2A
SCHEMBL844672 0.78 SLC6A4 (0.39) MEN1KMT2ALMNAHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 444 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12570675-B2 Boronic acid compounds LG CHEM, LTD. (KR) 2026-03-10 US disclosed
US-20250388615-A9 SUBSTITUTED 4-PHENYL PYRIDINE COMPOUNDS AS NON-SYSTEMIC TGR5 AGONISTS ARDELYX, INC. (US) 2025-12-25 US disclosed
EP-4561561-A2 SUBSTITUTED 3,4-DIHYDROQUINOLINONE INHIBITORS OF TSHR Septerna, Inc. (US) 2025-06-04 EP disclosed
US-20250066410-A1 SUBSTITUTED 4-PHENYL PYRIDINE COMPOUNDS AS NON-SYSTEMIC TGR5 AGONISTS ARDELYX, INC. (US) 2025-02-27 US disclosed
CN-119490464-A Preparation method of 1,2, 3-triazole compound and application thereof in antifungal field 中国人民解放军海军军医大学 2025-02-21 CN disclosed
WO-2025016469-A1 ALKOXY THIOPHENE ACYL ARYLAMINE COMPOUNDS AND USE THEREOF 复旦大学 2025-01-23 WO disclosed
CN-119320385-A Alkoxy thiophene carboxamide compounds and application thereof 复旦大学 2025-01-17 CN disclosed
EP-4474017-A2 NEW HETEROCYCLIC COMPOUNDS F. Hoffmann-La Roche AG (CH) 2024-12-11 EP disclosed
CN-118955358-A FXR partial agonist containing piperidine structure, and preparation method and application thereof 桂林医学院 2024-11-15 CN disclosed
US-12084472-B2 Substituted 4-phenyl pyridine compounds as non-systemic TGR5 agonists ARDELYX, INC. (US) 2024-09-10 US disclosed
US-5891889-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-04-06 US disclosed
WO-1997038665-A2 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-23 WO disclosed
US-5409943-A [(alkoxy)pyridinyl]amine compounds which are useful in the treatment of gastrointestinal disorders SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1995-04-25 US disclosed
EP-0625143-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1994-11-23 EP disclosed
WO-1993015055-A1 PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICINES SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1993-08-05 WO disclosed
WO-1993013092-A1 IMIDAZOLIDINEDIONE DERIVATIVES SARGES REINHARD (US) 1993-07-08 WO disclosed
US-5011840-A Imidazolidinedione derivatives in diabetes treatment PFIZER INC. (US) 1991-04-30 US disclosed
US-4698338-A ANTIBIOTICS ELI LILLY AND COMPANY (US) 1987-10-06 US disclosed
EP-0233780-A2 O-substituted oximino cephalosporins ELI LILLY AND COMPANY (US) 1987-08-26 EP disclosed
US-4077982-A HERBICIDES FMC CORPORATION (US) 1978-03-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250066410-A1 SUBSTITUTED 4-PHENYL PYRIDINE COMPOUNDS AS NON-SYSTEMIC TGR5 AGONISTS GPR119, GIPR, GLP1R TP53 4394/4885CYP3A4 448/4885IDO1 1111/4885
US-12570675-B2 Boronic acid compounds PSMB6, PSMB3, PSMB2 TP53 1120/4885CYP3A4 1946/4885IDO1 3016/4885
US-20250388615-A9 SUBSTITUTED 4-PHENYL PYRIDINE COMPOUNDS AS NON-SYSTEMIC TGR5 AGONISTS GPR119, GIPR, FFAR3 TP53 4523/4885CYP3A4 580/4885IDO1 1416/4885
US-12084472-B2 Substituted 4-phenyl pyridine compounds as non-systemic TGR5 agonists GPR119, GIPR, GLP1R TP53 4394/4885CYP3A4 448/4885IDO1 1111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.