D-Glutamate

D-Glutamate

SCHEMBL1899059

N[C@H](CCC(=O)O)C(=O)[O-].[K+]

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

AGTR1DHFRGABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTNR3C2PBP2XPTGS1PTGS2VKORC1blablaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAftsImrcAmrcBmrdApbp1apbp1bpbp2apbp2bpbp3polthyA

The experimentally established mechanism targets of D-Glutamate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP known ✓ O00591 2/20 0.50
GABRD known ✓ O14764 2/20 0.50
GABRA1 known ✓ P14867 2/20 0.50
GABRB1 known ✓ P18505 2/20 0.50
GABRG2 known ✓ P18507 2/20 0.50
GABRB3 known ✓ P28472 2/20 0.50
GABRA5 known ✓ P31644 2/20 0.50
GABRA3 known ✓ P34903 2/20 0.50
GABRA2 known ✓ P47869 2/20 0.50
GABRB2 known ✓ P47870 2/20 0.50
GABRA4 known ✓ P48169 2/20 0.50
GABRE known ✓ P78334 2/20 0.50
GABRA6 known ✓ Q16445 2/20 0.50
GABRG1 known ✓ Q8N1C3 2/20 0.50
GABRG3 known ✓ Q99928 2/20 0.50
GABRQ known ✓ Q9UN88 2/20 0.50
CYP1A2 P05177 2/20 0.62
GRM8 O00222 1/20 0.62
GRM6 O15303 1/20 0.62
GRIN2D O15399 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
D-Glutamate SCHEMBL82751 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL249807 1.00 CYP1A2 (0.62) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL4294624 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL10930916 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL1394398 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL11742429 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL2853216 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL11741892 0.98 CYP1A2 (0.60) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL10930108 0.96 CYP1A2 (0.58) CYP1A2GRM8GRM6GRIN2DGRIN3B
D-Glutamate SCHEMBL30787945 0.96 CYP1A2 (0.58) CYP1A2GRM8GRM6GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3395862-B1 RESIN COMPOSITION PELLETS MITSUBISHI CHEM CORP (JP) 2023-05-10 EP disclosed
EP-3281980-B1 RESIN COMPOSITION AND MULTILAYER STRUCTURE USING SAME, AND METHOD OF IMPROVING LONG-RUN STABILITY MITSUBISHI CHEM CORP (JP) 2021-03-03 EP disclosed
WO-2021015095-A1 PROTEIN PRODUCTION METHOD AND CELL-FREE PROTEIN SYNTHESIS KIT 大陽日酸株式会社 2021-01-28 WO disclosed
US-10611894-B2 Resin composition and multilayer structure using same, and method of improving long-run stability MITSUBISHI CHEMICAL CORPORATION (JP) 2020-04-07 US disclosed
US-10358533-B2 Resin composition pellet MITSUBISHI CHEMICAL CORPORATION (JP) 2019-07-23 US disclosed
US-20180371179-A1 RESIN COMPOSITION PELLET THE NIPPON SYNTHETIC CHEMICAL INDUSTRY CO., LTD. (JP) 2018-12-27 US disclosed
EP-3395862-A1 RESIN COMPOSITION PELLETS The Nippon Synthetic Chemical Industry Co., Ltd. (JP) 2018-10-31 EP disclosed
EP-2845881-B1 RESIN COMPOSITION, MELT FORMED ARTICLE, MULTILAYER STRUCTURE, AND PROCESS FOR PRODUCING RESIN COMPOSITION NIPPON SYNTHETIC CHEM IND CO LTD (JP) 2018-04-11 EP disclosed
US-20180044502-A1 RESIN COMPOSITION AND MULTILAYER STRUCTURE USING SAME, AND METHOD OF IMPROVING LONG-RUN STABILITY THE NIPPON SYNTHETIC CHEMICAL INDUSTRY CO., LTD. (JP) 2018-02-15 US disclosed
EP-3281980-A1 RESIN COMPOSITION AND MULTILAYER STRUCTURE USING SAME, AND METHOD OF IMPROVING LONG-RUN STABILITY The Nippon Synthetic Chemical Industry Co., Ltd. (JP) 2018-02-14 EP disclosed
US-5631294-A PHENOXY- OR PHENYL-ALKANOIC ACIDS BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631038-A COMPOUNDS (TASTANDS) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE ARE ADDED TO FOODS CONTAINING SODIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631295-A 2-(4-METHOXYPHENOXY)PROPIONIC ACID, TAURINE, ASPARTYLPHENYL ALANINE, ASPARTYLTYROSINE AND DIHYDROXYBENZOIC ACID BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631240-A KETONE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631299-A TAURINE OR AN ACCEPTABLE SALT (A TASTAND) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631252-A Specific eatable taste modifiers BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631232-A COMPOUNDS (TASTANDS-SUCH AS DERIVATIVES OF ASPARTIC ACID) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631231-A COMPOUNDS (TASTANDS, E.G., DIPEPTIDES) TO REDUCE OR ELIMINATE A BITTER OR METALLIC TASTE; FOODS; DRUGS; SWEETENERS; POTASSIUM CHLORIDE BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631272-A SUBSTITUTED TRYPTAMINES BIORESEARCH, INC. (US) 1997-05-20 US disclosed
US-5631292-A COMPOUNDS TO REMOVE BITTER TASTES FROM FOOD BIORESEARCH, INC. (US) 1997-05-20 US disclosed