SCHEMBL18992188

SCHEMBL18992188

O=C1C=C(O)C(=O)c2cc(Br)ccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 3/20 0.58
MCL1 Q07820 2/20 0.58
S100A4 P26447 2/20 0.57
PTPRC P08575 1/20 0.50
LCK P06239 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
ESR1 P03372 3/20 0.42
ESR2 Q92731 3/20 0.42
MAOA P21397 1/20 0.42
UGT1A1 P22309 1/20 0.42
MAOB P27338 1/20 0.42
BACE1 P56817 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
TGM2 P21980 1/20 0.39
CES1 P23141 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9389370 0.92 BCL2 (0.58) BCL2MCL1S100A4PTPRCLCK
SCHEMBL5817037 0.84 ESR2 (0.61) PTPRCCA1CA2CA7CA9
SCHEMBL29407366 0.84 ESR2 (0.61) PTPRCCA1CA2CA7CA9
SCHEMBL28845752 0.80 S100A4 (0.61) BCL2MCL1S100A4PTPRCLCK
SCHEMBL10086888 0.77 CA9 (0.44) CA1CA2CA7CA9ESR1
SCHEMBL30490 0.77 S100A4 (0.57) S100A4CA1CA2ESR1ESR2
SCHEMBL28591550 0.77 MAOA (0.53) BCL2MCL1LCKCA1CA2
SCHEMBL29404998 0.77 MAOA (0.53) BCL2MCL1LCKCA1CA2
SCHEMBL21013875 0.77 TGM2 (0.39) BCL2MCL1ESR1ESR2MAOA
SCHEMBL5811756 0.76 ESR2 (0.61) BCL2MCL1PTPRCCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10829427-B2 Naphthoquinones, pro-drugs, and methods of use thereof THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2020-11-10 US disclosed
US-10829427-B2 Naphthoquinones, pro-drugs, and methods of use thereof THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2020-11-10 US disclosed
US-20190071380-A1 NAPHTHOQUINONES, PRO-DRUGS, AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2019-03-07 US disclosed
US-20190071380-A1 NAPHTHOQUINONES, PRO-DRUGS, AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2019-03-07 US disclosed
WO-2017106624-A1 NAPTHOQUINONES, PRO-DRUGS, AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-06-22 WO disclosed
WO-2017106624-A1 NAPTHOQUINONES, PRO-DRUGS, AND METHODS OF USE THEREOF THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-06-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10829427-B2 Naphthoquinones, pro-drugs, and methods of use thereof NQO1, RECQL, ABCB1 BCL2 1184/4885MCL1 217/4885S100A4 2683/4885
US-20190071380-A1 NAPHTHOQUINONES, PRO-DRUGS, AND METHODS OF USE THEREOF NQO1, RECQL, ABCB1 BCL2 1184/4885MCL1 217/4885S100A4 2683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.