SCHEMBL1900363

SCHEMBL1900363

O=C1Cc2cc(-c3cccc(F)c3)ccc2N1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 5/20 0.68
CYP1A2 P05177 1/20 0.61
CYP11B1 P15538 1/20 0.61
CYP11B2 P19099 1/20 0.61
PDE3B Q13370 1/20 0.60
PDE3A Q14432 1/20 0.60
GRIA1 P42261 3/20 0.60
CACNG8 Q8WXS5 3/20 0.60
AHR P35869 2/20 0.50
PARP10 Q53GL7 1/20 0.50
PARP11 Q9NR21 1/20 0.50
OTUD7B Q6GQQ9 1/20 0.49
MAOB P27338 2/20 0.49
KIF11 P52732 1/20 0.49
TDP2 O95551 1/20 0.49
BRD4 O60885 1/20 0.48
CREBBP Q92793 1/20 0.48
ALOX5AP P20292 1/20 0.47
FEN1 P39748 1/20 0.47
PDK2 Q15119 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1897593 0.87 PDE3B (0.68) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL3309677 0.86 KIF11 (0.62) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL3132725 0.85 PGR (0.73) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL18189405 0.83 GRIA1 (0.70) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL152963 0.81 AHR (0.61) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL3519711 0.81 PGR (1.00) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL8263674 0.81 PGR (0.68) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL28203333 0.81 PGR (1.00) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL10714806 0.81 TDP2 (0.69) PGRCYP1A2CYP11B1CYP11B2PDE3B
SCHEMBL1900635 0.81 PDE3B (0.64) PGRCYP1A2CYP11B1CYP11B2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed