SCHEMBL1900635

SCHEMBL1900635

O=C1Cc2cc(-c3ccc(F)c(F)c3)ccc2N1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.64
PDE3A Q14432 1/20 0.64
PGR P06401 5/20 0.63
AHR P35869 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56
GRIA1 P42261 4/20 0.55
CACNG8 Q8WXS5 3/20 0.55
TDP2 O95551 3/20 0.51
KIF11 P52732 1/20 0.51
ALOX5AP P20292 1/20 0.49
FEN1 P39748 1/20 0.49
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
TNIK Q9UKE5 1/20 0.47
BMPR1B O00238 1/20 0.46
BMPR1A P36894 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1897593 0.86 PDE3B (0.68) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1908017 0.86 GRIA1 (0.62) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1896888 0.86 TDP2 (0.70) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1899619 0.83 PDE3B (0.56) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1900155 0.83 AHR (0.77) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL18189405 0.82 GRIA1 (0.70) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1902333 0.82 TDP2 (0.50) PDE3BPDE3APGRCYP1A2CYP11B1
SCHEMBL3132725 0.81 PGR (0.73) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL1900363 0.81 PGR (0.68) PDE3BPDE3APGRAHRCYP1A2
SCHEMBL24884440 0.80 GRIA1 (0.69) PDE3BPDE3APGRAHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed