SCHEMBL190042

SCHEMBL190042

COC(=O)C1CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.54
NPC1 O15118 1/20 0.54
FKBP1A P62942 1/20 0.52
LMNA P02545 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
POLB P06746 1/20 0.51
UCHL1 P09936 2/20 0.48
SCN4A P35499 1/20 0.48
EPHX2 P34913 1/20 0.48
USP30 Q70CQ3 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
KLK7 P49862 1/20 0.47
PEPD P12955 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1486184 1.00 HSD17B10 (0.58) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL883030 1.00 HSD17B10 (0.58) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
Hydrochloric Acid SCHEMBL29889454 0.98 HSD17B10 (0.57) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL2737884 0.95 FKBP1A (0.58) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL2898129 0.95 FKBP1A (0.58) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL88684 0.95 FKBP1A (0.58) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL6272597 0.94 HSD17B10 (0.60) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL3467497 0.94 HSD17B10 (0.60) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL6361642 0.94 HSD17B10 (0.60) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA
SCHEMBL18455416 0.94 FKBP1A (0.57) HSD17B10SMN1; SMN2NPC1FKBP1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 443 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4463455-B1 HETEROALICYCLIC DERIVATIVES AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SUVEN LIFE SCIENCES LTD (IN) 2026-04-29 EP disclosed
US-12391698-B2 Substituted piperidines and piperazines and methods for the treatment of CNS disorders SUVEN LIFE SCIENCES LIMITED (IN) 2025-08-19 US disclosed
US-20250186392-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF TENACIA BIOTECHNOLOGY HONG KONG CO LTD (HK) 2025-06-12 US disclosed
CN-119816491-A New spirocyclohexane derivatives, pharmaceutical compositions containing them and their use as anti-apoptotic inhibitors 法国施维雅药厂 2025-04-11 CN disclosed
CN-119775187-A Melanocortin-4 receptor agonists 株式会社LG化学 2025-04-08 CN disclosed
US-20250092049-A1 HETEROALICYCLIC DERIVATIVES AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SUVEN LIFE SCIENCES LIMITED (IN) 2025-03-20 US disclosed
WO-2025000265-A1 HETEROCYCLIC COMPOUNDS USEFULL AS SOS1 INHIBITOR SILEXON AI TECHNOLOGY CO., LTD. (CN) 2025-01-02 WO disclosed
US-20240425476-A1 2-(2,4,5-SUBSTITUTED-ANILINO)PYRIMIDINE COMPOUNDS ASTRAZENECA AB (SE) 2024-12-26 US disclosed
US-12167998-B2 Spiro-lactam NMDA receptor modulators and uses thereof TENACIA BIOTECHNOLOGY (HONG KONG) CO., LIMITED (CN) 2024-12-17 US disclosed
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2024-12-10 US disclosed
US-6756378-B2 BENZYL -UREA, -THIOUREA, OR -GUANIDINE DERIVATIVES THAT INHIBIT THE BINDING OF LIGANDS TO ALPHA 4 BETA 1 INTEGRIN (VLA-4) PHARMACOPEIA DRUG DISCOVERY, INC. 2004-06-29 US disclosed
WO-2004009599-A1 FIVE-MEMBERED HETEROAROMATIC OLEFINIC AZACYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS INHIBITORS OF NCOTINIC CHOLINERGIC RECEPTORS TARGACEPT, INC. (US) 2004-01-29 WO disclosed
EP-1317428-A1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-06-11 EP disclosed
US-20030078249-A1 VLA-4 inhibitor compounds DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-24 US disclosed
EP-1303485-A1 PYRROLIDINE DERIVATIVES AS INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
EP-1303507-A1 PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
US-20020160998-A1 Pharmaceutical compositions and methods for use TARGACEPT, INC. 2002-10-31 US disclosed
WO-2002006222-A1 PYRROLIDINE DERIVATIVES AS INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed
WO-2002006224-A1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed
WO-2002006271-A1 PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250186392-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN3A HSD17B10 2431/4885SMN1; SMN2 913/4885NPC1 1322/4885
US-12167998-B2 Spiro-lactam NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN3A HSD17B10 2431/4885SMN1; SMN2 913/4885NPC1 1322/4885
US-20030078249-A1 VLA-4 inhibitor compounds VCAM1, ICAM1, ITGA4 HSD17B10 3461/4885SMN1; SMN2 4151/4885NPC1 2939/4885
US-12391698-B2 Substituted piperidines and piperazines and methods for the treatment of CNS disorders GRIN2C, SLC1A2, CNR2 HSD17B10 2416/4885SMN1; SMN2 190/4885NPC1 129/4885
US-12162890-B2 Heteroaromatic NMDA receptor modulators and uses thereof GRIN2C, GRIN2A, GRIN1 HSD17B10 1332/4885SMN1; SMN2 4683/4885NPC1 2666/4885
US-20240425476-A1 2-(2,4,5-SUBSTITUTED-ANILINO)PYRIMIDINE COMPOUNDS EGFR, ERBB2, ERBB3 HSD17B10 4088/4885SMN1; SMN2 2671/4885NPC1 1895/4885
US-20250092049-A1 HETEROALICYCLIC DERIVATIVES AND THEIR USE IN THE TREATMENT OF CNS DISORDERS GRIN2C, CNR2, INA HSD17B10 593/4885SMN1; SMN2 238/4885NPC1 113/4885
US-20020160998-A1 Pharmaceutical compositions and methods for use AADAC, CYP3A7, CYP3A5 HSD17B10 483/4885SMN1; SMN2 4695/4885NPC1 273/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.