SCHEMBL1908017

SCHEMBL1908017

Cc1cc(-c2ccc3c(c2)CC(=O)N3)ccc1F

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 2/20 0.62
CACNG8 Q8WXS5 2/20 0.62
PDE3B Q13370 1/20 0.59
PDE3A Q14432 1/20 0.59
PGR P06401 4/20 0.58
DAPK3 O43293 1/20 0.54
NTRK1 P04629 1/20 0.54
PIM1 P11309 1/20 0.54
FLT3 P36888 1/20 0.54
GSK3B P49841 1/20 0.54
ROCK1 Q13464 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
AHR P35869 1/20 0.53
CYP1A2 P05177 1/20 0.52
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
CRBN Q96SW2 1/20 0.48
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4607881 0.87 KIF11 (0.61) GRIA1CACNG8PDE3BPDE3ADAPK3
SCHEMBL1900635 0.86 PDE3B (0.64) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL1897593 0.82 PDE3B (0.68) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL1896888 0.82 TDP2 (0.70) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL18189476 0.80 GRIA1 (0.82) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL27859220 0.80 PDE3B (0.64) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL1899619 0.79 PDE3B (0.56) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL1900155 0.79 AHR (0.77) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL18189405 0.78 GRIA1 (0.70) GRIA1CACNG8PDE3BPDE3APGR
SCHEMBL3132725 0.77 PGR (0.73) GRIA1CACNG8PDE3BPDE3APGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed