SCHEMBL19006771

SCHEMBL19006771

COc1cnc2n1-c1ccc(Br)cc1C(c1ccccn1)=NC2

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA3 P34903 11/20 0.66
GABRA2 P47869 8/20 0.66
GABRA1 P14867 8/20 0.66
GABRA5 P31644 7/20 0.66
GABRB2 P47870 5/20 0.66
ADRA1A P35348 2/20 0.47
TSHR P16473 1/20 0.46
GABRG2 P18507 7/20 0.39
GABRB3 P28472 7/20 0.39
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTR2A P28223 1/20 0.34
OPRK1 P41145 1/20 0.34
PDE4D Q08499 1/20 0.34
PTAFR P25105 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11828965 0.86 GABRA3 (0.73) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL29783033 0.86 GABRA3 (0.73) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL11732204 0.82 GABRA3 (0.64) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL11713247 0.81 GABRA3 (0.63) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL11834518 0.81 GABRA3 (0.63) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL11624016 0.80 GABRA1 (1.00) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL29385106 0.80 GABRA1 (1.00) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL11865356 0.79 GABRA1 (0.80) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL19006763 0.78 GABRA2 (0.47) GABRA3GABRA2GABRA1GABRA5GABRB2
SCHEMBL7311148 0.78 GABRA3 (0.70) GABRA3GABRA2GABRA1GABRA5GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017101808-A1 SHORT-ACTING BENZODIAZEPINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2017-06-22 WO disclosed