SCHEMBL19086466

SCHEMBL19086466

CON(C)C(=O)C1CC1=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 3/20 0.34
BCL2 P10415 1/20 0.34
SRD5A2 P31213 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1396157 0.82 MAPK1 (0.35) MCL1SRD5A2THRB
SCHEMBL1662468 0.79 MAPK1 (0.43) MCL1SRD5A2THRB
SCHEMBL870814 0.77 MCL1 (0.33) MCL1BCL2MEN1KMT2ATDP1
SCHEMBL2252786 0.72 MCL1 (0.33) MCL1BCL2MEN1KMT2ATDP1
SCHEMBL31352403 0.72 CRBN (0.39) MCL1BCL2SRD5A2
SCHEMBL1662124 0.71 THRB (0.39) MCL1BCL2SRD5A2THRB
SCHEMBL428708 0.70
SCHEMBL31623264 0.70 HSD11B1 (0.33) MCL1
SCHEMBL8532532 0.70 SRD5A2 (0.33) MCL1BCL2SRD5A2
SCHEMBL14895840 0.70 MCL1 (0.31) MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3189834-B1 USE OF GABAA RECEPTOR REINFORCING AGENT IN PREPARATION OF SEDATIVE AND ANESTHETIC MEDICAMENT HAISCO INNOVATIVE PHARMACEUTICAL PTE LTD (SG) 2024-01-17 EP disclosed
US-10729666-B2 Use of GABAA receptor reinforcing agent in preparation of sedative and anesthetic medicament HAISCO CHENGDU PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2020-08-04 US disclosed
US-20170290781-A1 USE OF GABAA RECEPTOR REINFORCING AGENT IN PREPARATION OF SEDATIVE AND ANESTHETIC MEDICAMENT HAISCO INNOVATIVE PHARMACEUTICAL PTE. LTD. (SG) 2017-10-12 US disclosed
EP-3189834-A1 USE OF GABAA RECEPTOR REINFORCING AGENT IN PREPARATION OF SEDATIVE AND ANESTHETIC MEDICAMENT Sichuan Haisco Pharmaceutical Co., Ltd. (CN) 2017-07-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10729666-B2 Use of GABAA receptor reinforcing agent in preparation of sedative and anesthetic medicament GABRA1, GABRA5, GABRA2 MCL1 4584/4885BCL2 4297/4885SRD5A2 1064/4885
US-20170290781-A1 USE OF GABAA RECEPTOR REINFORCING AGENT IN PREPARATION OF SEDATIVE AND ANESTHETIC MEDICAMENT GABRA1, GABRA5, GABRA2 MCL1 4584/4885BCL2 4297/4885SRD5A2 1064/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.