SCHEMBL19087047

SCHEMBL19087047

CNC(=O)CCn1cc(C)cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.60
LMNA P02545 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
GAA P10253 5/20 0.56
KMT2A Q03164 2/20 0.56
CYP3A4 P08684 2/20 0.53
CYP2C19 P33261 2/20 0.53
ALDH1A1 P00352 3/20 0.52
CYP1A2 P05177 2/20 0.52
MEN1 O00255 1/20 0.49
CYP2C9 P11712 1/20 0.49
PDK2 Q15119 2/20 0.46
ALPI P09923 1/20 0.44
ALPG P10696 1/20 0.44
PLAA Q9Y263 1/20 0.44
POLB P06746 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
BTK Q06187 1/20 0.38
KLKB1 P03952 1/20 0.38
PLK1 P53350 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10084730 0.84 ALPI (0.51) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL25976223 0.83 SMN1; SMN2 (0.56) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL28599036 0.82 PDK2 (0.45) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL10175541 0.81 LMNA (0.54) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL6937303 0.81 LMNA (0.54) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL19116732 0.81 HTT (0.45) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL19077855 0.81 PDK2 (0.44) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL18534152 0.80 LMNA (0.53) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL19087158 0.79 SMN1; SMN2 (0.52) HTTLMNASMN1; SMN2GAAKMT2A
SCHEMBL19087087 0.78 L3MBTL1 (0.56) HTTLMNASMN1; SMN2GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024097355-A1 DEUBIQUITINASE-TARGETING CHIMERAS AND RELATED METHODS VICINITAS THERAPEUTICS, INC. (US) 2024-05-10 WO disclosed
EP-3792256-A1 PYRIDINE AND PYRIDIMINE COMPOUNDS AS PI3K-GAMMA INHIBITORS Incyte Corporation (US) 2021-03-17 EP disclosed
EP-3400221-B1 PYRAZOL / IMIDAZOL SUBSTITUTED PYRIDINES AS PI3K-GAMMA INHIBITORS INCYTE CORP (US) 2020-08-26 EP disclosed
WO-2017120194-A1 PYRIDINE AND PYRIDIMINE COMPOUNDS AS PI3K-GAMMA INHIBITORS INCYTE CORPORATION (US) 2017-07-13 WO disclosed
US-20170190689-A1 PYRIDINE AND PYRIDIMINE COMPOUNDS AS PI3K-GAMMA INHIBITORS INCYTE CORPORATION 2017-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170190689-A1 PYRIDINE AND PYRIDIMINE COMPOUNDS AS PI3K-GAMMA INHIBITORS PIK3CG, PIK3CD, PIK3CB HTT 2012/4885LMNA 3680/4885SMN1; SMN2 1910/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.