SCHEMBL10175541

SCHEMBL10175541

Cc1cnn(CCC(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
GAA P10253 5/20 0.52
KMT2A Q03164 2/20 0.50
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
ALDH1A1 P00352 5/20 0.46
CYP1A2 P05177 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPK1 P28482 1/20 0.46
EGLN3 Q9H6Z9 1/20 0.46
MAPT P10636 1/20 0.46
KMO O15229 1/20 0.45
ALPI P09923 1/20 0.44
ALPG P10696 1/20 0.44
PLAA Q9Y263 1/20 0.44
PKM P14618 1/20 0.44
PDK2 Q15119 2/20 0.44
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28842191 0.98 LMNA (0.52) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL13127885 0.89 ALDH1A1 (0.50) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL12460554 0.88 SMN1; SMN2 (0.47) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL6937303 0.85 LMNA (0.54) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL19087158 0.84 SMN1; SMN2 (0.52) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL11983525 0.81 ALPI (0.54) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL18534152 0.81 LMNA (0.53) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL21576892 0.81 LMNA (0.50) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL18712865 0.81 LMNA (0.50) LMNAHTTSMN1; SMN2GAAKMT2A
SCHEMBL19087047 0.81 HTT (0.60) LMNAHTTSMN1; SMN2GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4029868-B1 MCL-1 INHIBITORS GILEAD SCIENCES INC (US) 2026-05-20 EP disclosed
WO-2024204554-A1 SPIROCYCLIC MORPHINAN DERIVATIVE 日本ケミファ株式会社 2024-10-03 WO disclosed
CN-117304130-A MCL-1 inhibitors 吉利德科学公司 2023-12-29 CN disclosed
US-20230312490-A1 MCL-1 INHIBITORS GILEAD SCIENCES, INC. 2023-10-05 US disclosed
US-11643400-B2 MCL-1 inhibitors GILEAD SCIENCES, INC. (US) 2023-05-09 US disclosed
US-20220340535-A1 MCL-1 INHIBITORS GILEAD SCIENCES, INC. 2022-10-27 US disclosed
EP-4029868-A1 MCL-1 INHIBITORS GILEAD SCIENCES, INC. (US) 2022-07-20 EP disclosed
EP-3793565-B1 MCL-1 INHIBITORS GILEAD SCIENCES INC (US) 2022-01-05 EP disclosed
WO-2021132524-A1 EPOXY AZEPAN DERIVATIVE 日本ケミファ株式会社 2021-07-01 WO disclosed
US-10988451-B2 MCL-1 inhibitors GILEAD SCIENCES, INC. (US) 2021-04-27 US disclosed
US-20130274240-A1 FLUORENE COMPOUND AND PHARMACEUTICAL USE THEREOF JAPAN TOBACCO INC (US) 2013-10-17 US disclosed
US-8466288-B2 Isoindolinone inhibitors of phosphatidylinositol 3-kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-18 US disclosed
US-8343994-B2 Fluorene compound and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2013-01-01 US disclosed
US-8343994-B2 Fluorene compound and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2013-01-01 US disclosed
US-20120040950-A1 ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-16 US disclosed
EP-2345629-A1 FLUORENE COMPOUND AND USE THEREOF FOR MEDICAL PURPOSES Japan Tobacco, Inc. (JP) 2011-07-20 EP disclosed
US-20100240634-A1 Fluorene Compound and Pharmaceutical Use Thereof JAPAN TOBACCO INC. (JP) 2010-09-23 US disclosed
US-20100240634-A1 Fluorene Compound and Pharmaceutical Use Thereof JAPAN TOBACCO INC. (JP) 2010-09-23 US disclosed
WO-2010041748-A1 FLUORENE COMPOUND AND USE THEREOF FOR MEDICAL PURPOSES 日本たばこ産業株式会社 (JP) 2010-04-15 WO disclosed
WO-2007002254-A2 BENZOCYCLOHEPTAPYRIDINES AS INHIBITORS OF THE RECEPTOR TYROSINE KINASE MET MERCK & CO., INC. (US) 2007-01-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240634-A1 Fluorene Compound and Pharmaceutical Use Thereof FH, PCK2, PC LMNA 527/4885HTT 1111/4885SMN1; SMN2 518/4885
US-20230312490-A1 MCL-1 INHIBITORS MCL1, BCL2L1, BCL2 LMNA 1458/4885HTT 2323/4885SMN1; SMN2 1771/4885
US-20120040950-A1 ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE PIK3CD, PIK3CA, PIK3R5 LMNA 2298/4885HTT 1061/4885SMN1; SMN2 1801/4885
US-11643400-B2 MCL-1 inhibitors MCL1, BCL2L1, BCL2 LMNA 1458/4885HTT 2323/4885SMN1; SMN2 1771/4885
US-20130274240-A1 FLUORENE COMPOUND AND PHARMACEUTICAL USE THEREOF FH, PCK2, PC LMNA 527/4885HTT 1111/4885SMN1; SMN2 518/4885
US-10988451-B2 MCL-1 inhibitors MCL1, BCL2L1, BCL2 LMNA 1458/4885HTT 2323/4885SMN1; SMN2 1771/4885
US-20220340535-A1 MCL-1 INHIBITORS MCL1, BCL2L1, BCL2 LMNA 1458/4885HTT 2323/4885SMN1; SMN2 1771/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.