SCHEMBL19087096

SCHEMBL19087096

Fc1c(C(F)(F)F)c(C(F)(F)F)nn1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.42
PTGS2 P35354 4/20 0.42
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP11B2 P19099 1/20 0.36
BRAF P15056 1/20 0.35
CYP2D6 P10635 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16769783 0.88 PTGS1 (0.40) PTGS1PTGS2NPSR1SMN1; SMN2POLB
SCHEMBL15060859 0.84 PTGS1 (0.37) PTGS1PTGS2NPSR1TDP1SMN1; SMN2
SCHEMBL12609497 0.82 PTGS1 (0.35) PTGS1PTGS2CYP1A2CYP2C9MEN1
SCHEMBL19087157 0.81 CYP1A2 (0.47) PTGS1NPSR1TDP1SMN1; SMN2POLB
SCHEMBL29248058 0.79 POLB (0.50) PTGS1PTGS2NPSR1TDP1SMN1; SMN2
SCHEMBL13860574 0.77 NPC1 (0.47) PTGS1PTGS2CYP1A2CYP2C9CYP2C19
SCHEMBL28604457 0.77 ALDH1A1 (0.42) PTGS1PTGS2NPSR1TDP1SMN1; SMN2
SCHEMBL3382151 0.77 PTGS2 (0.44) PTGS1PTGS2LMNAHTT
SCHEMBL3384424 0.77 PTGS1 (0.39) PTGS1PTGS2NPSR1TDP1SMN1; SMN2
SCHEMBL3379848 0.77 CACNA1G (0.39) PTGS1PTGS2SMN1; SMN2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9957256-B2 Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-05-01 US disclosed
US-9845312-B2 Process for the preparation of 5-fluoro-1H-pyrazoles BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-12-19 US disclosed
US-20170233348-A1 Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene ELANCO ANIMAL HEALTH GMBH (DE) 2017-08-17 US disclosed
US-9725415-B2 Process for the preparation of 5-fluoro-1H-pyrazoles BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2017-08-08 US disclosed
US-20170190690-A1 Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene ELANCO ANIMAL HEALTH GMBH (DE) 2017-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233348-A1 Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene CYP2F1, CYP4F2, CYP4F11 PTGS1 2843/4885PTGS2 3363/4885NPSR1 2674/4885
US-20170190690-A1 Process for the preparation of 5-fluoro-1H-pyrazoles starting from hexafluoropropene CYP2F1, CYP4F2, CYP4F11 PTGS1 2843/4885PTGS2 3363/4885NPSR1 2674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.