SCHEMBL19142147

SCHEMBL19142147

Cc1cccc(S)c1NN

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
ACHE P22303 1/20 0.39
GAA P10253 1/20 0.38
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
CYP1A2 P05177 2/20 0.35
CYP2A6 P11509 1/20 0.35
CD44 P16070 1/20 0.34
ALDH1A1 P00352 3/20 0.34
PSMD14 O00487 1/20 0.34
COPS5 Q92905 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1289385 0.83 GAA (0.44) TSHRACHEGAAGRIN2DGRIN3B
Hydrochloric Acid SCHEMBL1457203 0.80 CYP3A4 (0.48) TSHRACHEGAAGRIN2DGRIN3B
SCHEMBL14610527 0.77 TSHR (0.39) TSHRACHEGRIN2DGRIN3BGRIN1
SCHEMBL23030132 0.74 CD44 (0.52) TSHRACHEGAAGRIN2DGRIN3B
SCHEMBL21733184 0.74 CYP3A4 (0.36) TSHRCD44ALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL10522290 0.74 DRD2 (0.47) GAAGRIN2DGRIN3BGRIN1GRIN2A
Methylamine SCHEMBL27412030 0.73 CYP3A4 (0.46) TSHRACHECYP1A2CYP2A6CD44
SCHEMBL21876495 0.73 ACHE (0.48) TSHRACHEGAAGRIN2DGRIN3B
SCHEMBL1997895 0.73 GAA (0.59) GAAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL28057157 0.73 TRPA1 (0.50) TSHRGAAGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046799-B1 PHOSPHOINOSITIDE 3-KINASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GENENTECH INC (US) 2017-07-19 EP disclosed