SCHEMBL19198136

SCHEMBL19198136

Fc1ccccc1CNc1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
CYP1A2 P05177 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HPGD P15428 1/20 0.53
LTA4H P09960 1/20 0.51
RAB9A P51151 1/20 0.51
KCNH3 Q9ULD8 1/20 0.51
MAPT P10636 2/20 0.50
GSK3B P49841 2/20 0.50
ATM Q13315 1/20 0.50
PLA2G1B P04054 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
ATG4B Q9Y4P1 1/20 0.50
CDC7 O00311 1/20 0.50
PLK4 O00444 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3906088 0.85 TAAR1 (0.50) KMT2ALTA4HRAB9AMETAP2SGMS2
SCHEMBL11060955 0.80 LTA4H (0.51) ALDH1A1LTA4HRAB9AGSK3BKDM4E
SCHEMBL30520309 0.80 KDM4E (0.59) KMT2AMEN1L3MBTL1ALDH1A1HPGD
SCHEMBL3254598 0.80 KDM4E (0.59) KMT2AMEN1L3MBTL1ALDH1A1HPGD
SCHEMBL11513654 0.80 KMT2A (0.72) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL19197793 0.78 KDM4C (0.61) KMT2ACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL19198153 0.78 ALDH1A1 (0.64) KMT2AMEN1CYP2C9ALDH1A1LTA4H
SCHEMBL25415696 0.76 RAB9A (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD
SCHEMBL22191674 0.76 L3MBTL1 (0.53) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL30520324 0.76 RAB9A (0.51) CYP1A2CYP2C9CYP2C19ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11214542-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2022-01-04 US disclosed
US-20210009520-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-01-14 US disclosed
US-10807956-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-10-20 US disclosed
US-20200172485-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-06-04 US disclosed
US-10597365-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-03-24 US disclosed
US-20190077758-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-03-14 US disclosed
US-10179769-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-15 US disclosed
US-20180044296-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2018-02-15 US disclosed
US-20170298025-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2017-10-19 US disclosed
US-9725441-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2017-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190077758-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-11214542-B2 Histone demethylase inhibitors KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-20170298025-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-10179769-B2 Histone demethylase inhibitors KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-10807956-B2 Histone demethylase inhibitors KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-20180044296-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-20210009520-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-20200172485-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885
US-10597365-B2 Histone demethylase inhibitors KDM1B, KDM5A, KDM1A KMT2A 45/4885MEN1 1315/4885CYP1A2 1445/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.