SCHEMBL1920221

SCHEMBL1920221

O=C(O)C(c1cc(F)ccc1S(=O)(=O)N(CC(=O)N1CCCC1c1ccccc1)c1ccc(Cl)cc1)N(c1ccc(Cl)cc1)S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
MDM4 O15151 1/20 0.39
MDM2 Q00987 1/20 0.39
LMNA P02545 3/20 0.37
PSEN1 P49768 7/20 0.37
PSEN2 P49810 7/20 0.37
APH1B Q8WW43 7/20 0.37
NCSTN Q92542 7/20 0.37
APH1A Q96BI3 7/20 0.37
PSENEN Q9NZ42 7/20 0.37
UTS2R Q9UKP6 2/20 0.37
HSD11B1 P28845 1/20 0.36
ALDH1A1 P00352 1/20 0.35
POLB P06746 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920502 0.93 LMNA (0.41) CRHBPCRHR2LMNAPSEN1PSEN2
SCHEMBL1920213 0.90 KMT2A (0.41) CRHBPCRHR2LMNAPSEN1PSEN2
SCHEMBL1921822 0.89 MDM4 (0.40) CRHBPCRHR2MDM4MDM2LMNA
SCHEMBL1920294 0.89 MDM4 (0.48) CRHBPCRHR2MDM4MDM2LMNA
SCHEMBL1920212 0.88 CRHBP (0.44) CRHBPCRHR2MDM4MDM2LMNA
SCHEMBL1920350 0.88 MAPT (0.43) MDM4MDM2LMNAALDH1A1POLB
SCHEMBL1919880 0.88 MDM4 (0.39) CRHBPCRHR2MDM4MDM2PSEN1
SCHEMBL1919721 0.88 CRHBP (0.38) CRHBPCRHR2MDM4MDM2LMNA
SCHEMBL3422507 0.86 CRHBP (0.51) CRHBPCRHR2LMNAPSEN1PSEN2
SCHEMBL1630642 0.86 CRHBP (0.51) CRHBPCRHR2LMNAPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245006-B1 SULFONAMIDES AS OREXIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-01 EP disclosed