SCHEMBL1920294

SCHEMBL1920294

COc1ccc(S(=O)(=O)N(c2ccc(Cl)cc2)C(C(=O)O)c2cc(OC)ccc2S(=O)(=O)N(CC(=O)N2CCCC2c2ccc(F)cc2)c2ccc(Cl)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM4 O15151 1/20 0.48
MDM2 Q00987 1/20 0.48
MAPT P10636 7/20 0.41
TP53 P04637 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
OXTR P30559 3/20 0.39
AVPR1A P37288 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
ALDH1A1 P00352 2/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920366 0.97 MDM4 (0.42) MDM4MDM2MAPTOXTRAVPR1A
SCHEMBL1920350 0.94 MAPT (0.43) MDM4MDM2MAPTOXTRAVPR1A
SCHEMBL1920212 0.94 CRHBP (0.44) MDM4MDM2MAPTTP53CRHBP
SCHEMBL1919930 0.92 MDM4 (0.39) MDM4MDM2MAPTOXTRAVPR1A
SCHEMBL1921822 0.92 MDM4 (0.40) MDM4MDM2MAPTTP53CRHBP
SCHEMBL1919944 0.92 CRHBP (0.47) MDM4MDM2MAPTTP53CRHBP
SCHEMBL1919880 0.91 MDM4 (0.39) MDM4MDM2MAPTCRHBPCRHR2
SCHEMBL1920870 0.90 OXTR (0.46) MAPTOXTRAVPR1ANPSR1ALDH1A1
SCHEMBL1920825 0.90 KMT2A (0.45) MDM4MDM2MAPTOXTRAVPR1A
SCHEMBL1920685 0.89 KMT2A (0.41) MDM4MDM2MAPTOXTRAVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245006-B1 SULFONAMIDES AS OREXIN ANTAGONISTS HOFFMANN LA ROCHE (CH) 2011-06-01 EP disclosed