SCHEMBL1921249

SCHEMBL1921249

N#Cc1ncc(OCc2ccccc2)cc1OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.53
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
XDH P47989 1/20 0.44
MAPT P10636 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RAB9A P51151 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
IMPDH2 P12268 1/20 0.43
ALOX5 P09917 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25387499 0.85 XDH (0.47) MAOBXDHSMN1; SMN2HTTLMNA
SCHEMBL16740400 0.84 CSF1R (0.47) MAOBPDGFRBPDGFRAMAPTMEN1
SCHEMBL12985052 0.84 GCK (0.48) MAOBXDHMAPTMEN1KMT2A
SCHEMBL20607927 0.84 GCK (0.46) MAOBXDHSMN1; SMN2HTTSTAT3
SCHEMBL1675480 0.84 MAOB (0.51) MAOBPDGFRBPDGFRAMAPTHSD17B10
SCHEMBL18865570 0.84 PLAU (0.54) MAOBXDHSMN1; SMN2HTTRAB9A
SCHEMBL25390493 0.80 PPIA (0.39) MAOBXDHMAPTMEN1KMT2A
SCHEMBL31662431 0.77 MAOB (0.51) MAOBMAPTHSD17B10MEN1KMT2A
SCHEMBL7248256 0.77 ALDH1A1 (0.50) MAOBXDHMAPTSMN1; SMN2LMNA
SCHEMBL4214379 0.76 LTA4H (0.58) MAOBMAPTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 81 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2022-08-30 US claimed
US-20210137901-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2021-05-13 US claimed
EP-4698520-A1 RAF-MEK PROTEIN COMPLEX MODULATORS AND METHODS OF USE THEREOF Gandeeva Therapeutics, Inc. (US) 2026-02-25 EP disclosed
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2025-11-25 US disclosed
CN-116472266-B Compounds as prolyl hydroxylase inhibitors and methods of making the same 苏中药业集团股份有限公司 2025-05-30 CN disclosed
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE WARNER CHILCOTT COMPANY, LLC (PR) 2024-10-31 US disclosed
WO-2024220708-A1 RAF-MEK PROTEIN COMPLEX MODULATORS AND METHODS OF USE THEREOF GANDEEVA THERAPEUTICS, INC. (US) 2024-10-24 WO disclosed
WO-2024079708-A1 A PROCESS FOR THE PREPARATION OF VADADUSTAT OR SALTS THEREOF AMI LIFESCIENCES PRIVATE LIMITED (IN) 2024-04-18 WO disclosed
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2024-01-30 US disclosed
EP-3888658-B1 EIF4-A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO EFFECTOR THERAPEUTICS INC (US) 2023-12-27 EP disclosed
US-20230295179-A1 EIF4A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO EFFECTOR THERAPEUTICS, INC. 2023-09-21 US disclosed
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
US-20100331374-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE AKEBIA THERAPEUTICS, INC. 2010-12-30 US disclosed
EP-2044005-B1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE WARNER CHILCOTT CO LLC (PR) 2010-10-20 EP disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
EP-2044005-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE The Procter and Gamble Company (US) 2009-04-08 EP disclosed
WO-2008002576-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-20230295179-A1 EIF4A-INHIBITING COMPOUNDS AND METHODS RELATED THERETO EIF4A1, EIF4A2, EIF4A3 MAOB 3586/4885PDGFRB 2340/4885PDGFRA 1895/4885
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, EGLN2 MAOB 349/4885PDGFRB 107/4885PDGFRA 104/4885
US-20100331374-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-20210137901-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885
US-20100331303-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A MAOB 461/4885PDGFRB 109/4885PDGFRA 130/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.