SCHEMBL1922533

SCHEMBL1922533

O=[N+]([O-])c1ccc(Cl)c(Cl)c1-c1ccc[c]c1Oc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.44
MEN1 O00255 1/20 0.44
TTR P02766 1/20 0.44
ALB P02768 1/20 0.44
THRB P10828 1/20 0.44
KMT2A Q03164 1/20 0.44
PIN1 Q13526 2/20 0.41
HPGD P15428 1/20 0.35
MAPK8 P45983 1/20 0.35
MAPT P10636 5/20 0.34
POLB P06746 2/20 0.34
APEX1 P27695 1/20 0.34
CASP6 P55212 1/20 0.34
ALDH1A1 P00352 3/20 0.33
VCAM1 P19320 2/20 0.33
S100A4 P26447 2/20 0.33
MERTK Q12866 1/20 0.33
PTPRC P08575 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11145042 0.76 PIN1 (0.46) TDP1MEN1TTRALBTHRB
SCHEMBL1922535 0.75 TDP1 (0.43) TDP1MEN1TTRALBTHRB
SCHEMBL11069630 0.73 TDP1 (0.57) TDP1MEN1TTRALBTHRB
SCHEMBL11996397 0.73 TDP1 (0.48) TDP1MEN1TTRALBTHRB
SCHEMBL28619341 0.70 TDP1 (0.58) TDP1MEN1TTRALBTHRB
SCHEMBL8123617 0.70 PDE7A (0.43) TDP1MEN1TTRALBTHRB
SCHEMBL6036733 0.68 LTA4H (0.42) MEN1KMT2AMAPTPOLBALDH1A1
SCHEMBL2533674 0.67 LTA4H (0.41) TDP1MEN1KMT2AMAPTALDH1A1
SCHEMBL5392376 0.67 LTA4H (0.41) TDP1MEN1KMT2AHPGDALDH1A1
SCHEMBL10883530 0.66 TDP1 (0.71) TDP1MEN1TTRALBTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981854-B1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-06-01 EP disclosed