SCHEMBL19249079

SCHEMBL19249079

Oc1ccccc1COc1cc(Br)cc2[nH]ncc12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 12/20 0.45
TDO2 P48775 11/20 0.44
PKM P14618 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC6A4 P31645 1/20 0.35
HTR6 P50406 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19249080 0.85 IDO1 (0.51) IDO1TDO2SLC6A4HTR6
SCHEMBL19249340 0.77 PTGER1 (0.37) IDO1TDO2MAPTMAPK1NPSR1
SCHEMBL19249341 0.76 IDO1 (0.42) IDO1TDO2MAPTSMN1; SMN2MAPK1
SCHEMBL28449826 0.75 TDO2 (0.67) IDO1TDO2PKMMAPTMEN1
SCHEMBL17440906 0.74 IDO1 (0.51) IDO1TDO2
SCHEMBL19249082 0.73 RXRA (0.48) IDO1TDO2NPC1RAB9ASMN1; SMN2
SCHEMBL19248989 0.73 MRGPRX4 (0.53) IDO1TDO2MEN1KMT2ANPC1
SCHEMBL17440928 0.72 MAOB (0.45) IDO1TDO2MAPTMEN1KMT2A
SCHEMBL19248986 0.71 CCR5 (0.48) IDO1TDO2MAPTMEN1KMT2A
SCHEMBL19249081 0.71 MAPT (0.46) IDO1TDO2PKMMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133258-A1 1H-INDAZOLE DERIVATIVE AND USE THEREOF AS IDO INHIBITOR 西华大学 2017-08-10 WO disclosed