SCHEMBL19257727

SCHEMBL19257727

CCC(CC(C)C(=O)O)c1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
ENPEP Q07075 2/20 0.37
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996178 0.85 ESR1 (0.51) HDAC8HDAC6AKR1C3AKR1C2TDP1
SCHEMBL12191565 0.84 APAF1 (0.50) POLBAPAF1ALDH1A1LMNA
SCHEMBL22267938 0.83 HDAC8 (0.41) HDAC8HDAC6ADRA2AADRA2BADRA2C
SCHEMBL19257724 0.81 GRIA4 (0.41) HDAC8HDAC6ENPEPAKR1C3AKR1C2
SCHEMBL13418590 0.80 NR1I2 (0.38) HDAC8HDAC6AKR1C3AKR1C2SMN1; SMN2
SCHEMBL19199258 0.78 ADRA2A (0.40) HDAC8HDAC6ADRA2AADRA2BADRA2C
SCHEMBL10429251 0.77 LMNA (0.50) POLBSMN1; SMN2ALDH1A1LMNA
SCHEMBL12384004 0.77 GRIA4 (0.39) HDAC8HDAC6ADRA2AADRA2BADRA2C
SCHEMBL13418600 0.75 APAF1 (0.45) APAF1LMNACYP1A2
SCHEMBL22267939 0.75 ALDH1A1 (0.38) HDAC8HDAC6ENPEPAKR1C3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017134547-A1 TUBULYSIN ANALOGS AND METHODS FOR THEIR PREPARATION PFIZER INC. (US) 2017-08-10 WO disclosed