SCHEMBL19258560

SCHEMBL19258560

Nc1nc(-n2ncc3ncc(C(F)(F)F)cc32)ncc1F

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 14/20 0.34
GRIN2B Q13224 14/20 0.34
CYP11B2 P19099 2/20 0.34
CYP11B1 P15538 1/20 0.34
MAT2A P31153 1/20 0.32
XDH P47989 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19258476 0.84 GRIN1 (0.33) GRIN1GRIN2B
SCHEMBL19250590 0.82 GRIN1 (0.34) GRIN1GRIN2B
SCHEMBL19258556 0.79 MAP3K14 (0.30)
SCHEMBL19259012 0.74 MEN1 (0.32) GRIN2B
SCHEMBL19258499 0.71 PDE10A (0.34)
SCHEMBL19259135 0.69 RPS6KA5 (0.37) GRIN2B
SCHEMBL19258987 0.65 GRIN1 (0.35) GRIN1GRIN2BCYP11B2
SCHEMBL119201 0.63 ALDH1A1 (0.43) CYP11B2CYP11B1ALDH1A1
Bromide SCHEMBL6033070 0.62 ALDH1A1 (0.42) CYP11B2CYP11B1ALDH1A1
SCHEMBL19258966 0.61 ALDH1A1 (0.35) GRIN1GRIN2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed