SCHEMBL19258966

SCHEMBL19258966

C=C(C)n1ncc2ncc(C(F)(F)F)cc21

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
AGBL2 Q5U5Z8 1/20 0.34
GRIN1 Q05586 14/20 0.34
GRIN2B Q13224 14/20 0.34
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19258971 0.68 RPS6KA5 (0.36) ALDH1A1KDM4E
SCHEMBL24695579 0.64 AGBL2 (0.46) ALDH1A1KDM4EAGBL2GAA
SCHEMBL30231011 0.63 CA12 (0.41) ALDH1A1KDM4EHTT
SCHEMBL19259003 0.61 HDAC8 (0.38) KDM4EPOLB
SCHEMBL27284155 0.61 ALDH1A1 (0.63) ALDH1A1KDM4EPOLBGAAHTT
SCHEMBL19258560 0.61 GRIN1 (0.34) ALDH1A1GRIN1GRIN2B
SCHEMBL11631751 0.60 HRH4 (0.39) ALDH1A1KDM4EPOLBPKMAGBL2
SCHEMBL24609261 0.60 ALDH1A1 (0.31) ALDH1A1KDM4EGRIN1GRIN2B
SCHEMBL18366009 0.60 ALDH1A1 (0.39) ALDH1A1KDM4EAGBL2HTT
SCHEMBL21730132 0.59 ALDH1A1 (0.42) ALDH1A1KDM4EPOLBPKMAGBL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed