SCHEMBL19258951

SCHEMBL19258951

C=C(C)n1ncc2ncc(F)cc21

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 9/20 0.33
GRIN1 Q05586 8/20 0.33
MT-CO1 P00395 1/20 0.32
MT-CO2 P00403 1/20 0.32
EDNRA P25101 1/20 0.32
OPRM1 P35372 1/20 0.32
HTR2B P41595 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19258966 0.80 ALDH1A1 (0.35) GRIN2BGRIN1
SCHEMBL33527364 0.73 GRIN1 (0.36) GRIN2BGRIN1MT-CO1MT-CO2EDNRA
SCHEMBL19258971 0.71 RPS6KA5 (0.36)
SCHEMBL19258987 0.67 GRIN1 (0.35) GRIN2BGRIN1
SCHEMBL19259003 0.64 HDAC8 (0.38)
SCHEMBL19630106 0.61 PIK3CB (0.41) GRIN2BGRIN1
SCHEMBL29640181 0.61 ELANE (0.41)
SCHEMBL23544518 0.58
SCHEMBL30621458 0.58 ALDH1A1 (0.39) GRIN2BGRIN1
SCHEMBL19231295 0.58 KCNH2 (0.39) GRIN2BGRIN1MT-CO1MT-CO2EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed