SCHEMBL19259003

SCHEMBL19259003

C=C(C)n1ncc2nc(C)ccc21

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.38
CHEK1 O14757 1/20 0.34
AURKA O14965 1/20 0.34
DAPK3 O43293 1/20 0.34
CSNK1A1 P48729 1/20 0.34
GSK3A P49840 1/20 0.34
LIMK1 P53667 1/20 0.34
IKBKE Q14164 1/20 0.34
MAPK14 Q16539 1/20 0.34
TAOK1 Q7L7X3 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
CYP1A2 P05177 3/20 0.33
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
CASP6 P55212 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14299249 0.83 CHEK1 (0.51) HDAC8CHEK1AURKADAPK3CSNK1A1
SCHEMBL19258971 0.72 RPS6KA5 (0.36) KDM4E
SCHEMBL7927906 0.72 HDAC8 (0.39) HDAC8CYP1A2KDM4ELMNAPOLB
SCHEMBL19258951 0.64 GRIN2B (0.33)
SCHEMBL10124285 0.63 NR3C1 (0.50) CYP1A2
SCHEMBL19258966 0.61 ALDH1A1 (0.35) KDM4EPOLB
SCHEMBL15345018 0.60 ALOX15 (0.50) HDAC8LMNA
SCHEMBL7512293 0.60 CYP1A2 (0.59) CYP1A2KDM4ELMNAPOLBCASP6
SCHEMBL21241066 0.59
SCHEMBL21874171 0.59 CHEK1 (0.41) HDAC8CHEK1AURKADAPK3CSNK1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed