SCHEMBL19259983

SCHEMBL19259983

[CH2]c1ccc(S(=O)(=O)c2ccc(-c3ccccc3)c(S(C)(=O)=O)c2)s1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 10/20 0.68
LOX P28300 8/20 0.57
MAOA P21397 5/20 0.57
KCNH2 Q12809 3/20 0.45
LOXL3 P58215 1/20 0.43
AOC3 Q16853 1/20 0.43
PTGS2 P35354 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19274325 0.81 LOXL2 (1.00) LOXL2LOXMAOAKCNH2LOXL3
Hydrochloric Acid SCHEMBL19259892 0.80 LOXL2 (1.00) LOXL2LOXMAOAKCNH2LOXL3
SCHEMBL28646852 0.73 LOX (0.66) LOXL2LOXMAOAKCNH2LOXL3
SCHEMBL19274305 0.73 LOX (1.00) LOXL2LOXMAOAKCNH2LOXL3
SCHEMBL28644342 0.72 LOXL2 (0.63) LOXL2LOXMAOAKCNH2LOXL3
SCHEMBL11045136 0.68 PTGS2 (0.53) LOXL2LOXMAOAPTGS2
SCHEMBL1368722 0.67 LOXL2 (0.47) LOXL2LOXMAOAPTGS2
SCHEMBL6303182 0.67 LOXL2 (0.50) LOXL2LOXMAOAKCNH2PTGS2
SCHEMBL27765267 0.67 ALOX5 (0.55) LOXL2PTGS2
SCHEMBL3464178 0.67 LOX (0.44) LOXL2LOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3416956-A1 METHYLAMINE DERIVATIVES AS LYSYSL OXIDASE INHIBITORS FOR THE TREATMENT OF CANCER The Institute of Cancer Research : The Royal Cancer Hospital (GB) 2018-12-26 EP disclosed
WO-2017141049-A1 METHYLAMINE DERIVATIVES AS LYSYSL OXIDASE INHIBITORS FOR THE TREATMENT OF CANCER THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (GB) 2017-08-24 WO disclosed